SCHEMBL8550771

SCHEMBL8550771

CC(C)Sc1cccc(NC(=O)Nc2ccc3scc(C4CCN(C(C)C)CC4)c3c2)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.40
EPHX2 P34913 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
KDR P35968 5/20 0.35
MEN1 O00255 2/20 0.35
MAPT P10636 2/20 0.35
KMT2A Q03164 2/20 0.35
TP53 P04637 1/20 0.35
POLB P06746 1/20 0.35
MAPK1 P28482 1/20 0.35
HSD17B10 Q99714 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
KCNJ6 P48051 1/20 0.35
KCNJ3 P48549 1/20 0.35
ITGB2 P05107 1/20 0.34
ICAM1 P05362 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8548440 0.86 CA2 (0.43) ALDH1A1EPHX2KDRMEN1KMT2A
SCHEMBL7486039 0.82 HTR1D (0.53) DRD2
SCHEMBL8549413 0.82 ALDH1A1 (0.40) ALDH1A1EPHX2SMN1; SMN2MEN1MAPT
SCHEMBL8704365 0.78 DRD2 (0.42) ALDH1A1EPHX2SMN1; SMN2MEN1MAPT
SCHEMBL8708863 0.78 UBE2M (0.47) UBE2MDCUN1D1
SCHEMBL8551242 0.76 MEN1 (0.43) MEN1MAPTKMT2ACYP1A2CYP3A4
SCHEMBL8548444 0.76 ALDH1A1 (0.39) ALDH1A1TP53HRH3DRD2SLC6A4
SCHEMBL8552303 0.75 RAB9A (0.43) SMN1; SMN2TP53HRH3
SCHEMBL8547892 0.74 HTR1D (0.46) HRH3
SCHEMBL8547952 0.73 HTR1D (0.45) ALDH1A1SMN1; SMN2HSD17B10CYP3A4HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5792763-A MIGRAINES; ANALGESICS; DISEASES LINKED TO DECREASED NEUROTRANMISSION OF SEROTONIN IN MAMMALS ELI LILLY AND COMPANY (US) 1998-08-11 US disclosed
WO-1998015545-A1 NEW SEROTONIN 5-HT1F AGONISTS ELI LILLY AND COMPANY (US) 1998-04-16 WO disclosed
EP-0835869-A2 New serotonin 5-HT1F agonists ELI LILLY AND COMPANY (US) 1998-04-15 EP disclosed