SCHEMBL8550982

SCHEMBL8550982

CCOC(=O)Oc1[nH]c2cc(OCc3ccccc3)c(OC)cc2c1-c1ccc(OC)cc1OCC(=O)O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSV O60911 2/20 0.44
CTSL P07711 2/20 0.44
SRD5A1 P18405 1/20 0.42
SRD5A2 P31213 1/20 0.42
PTPN1 P18031 3/20 0.41
FFAR1 O14842 4/20 0.40
PPARD Q03181 2/20 0.38
TUBB4A P04350 1/20 0.38
TUBB P07437 1/20 0.38
TUBA3C P0DPH7 1/20 0.38
TUBA1B P68363 1/20 0.38
TUBA4A P68366 1/20 0.38
TUBB4B P68371 1/20 0.38
TUBB3 Q13509 1/20 0.38
TUBB2A Q13885 1/20 0.38
TUBB8 Q3ZCM7 1/20 0.38
TUBA3E Q6PEY2 1/20 0.38
TUBA1A Q71U36 1/20 0.38
TUBA1C Q9BQE3 1/20 0.38
TUBB6 Q9BUF5 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8591475 0.93 PTPN1 (0.42) PTPN1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL8553723 0.90 FFAR1 (0.44) CTSVCTSLPTPN1FFAR1PPARD
SCHEMBL8552525 0.88 ELANE (0.38) PTPN1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL8553299 0.87 PTPN1 (0.38) PTPN1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL8553319 0.85 PDE4B (0.40) PTPN1ELANEALDH1A1MAPTHPGD
SCHEMBL8551848 0.79 CTSV (0.52) CTSVCTSLSRD5A1SRD5A2TUBB4A
SCHEMBL8697633 0.79 POLB (0.37) SRD5A1SRD5A2PTPN1HDAC8
SCHEMBL8697275 0.77 PTPN1 (0.42) PTPN1ALDH1A1MAPT
SCHEMBL8553266 0.76 EDNRB (0.56) CTSVCTSLSRD5A1SRD5A2ALDH1A1
SCHEMBL8546890 0.74 EDNRB (0.44) CTSVCTSLSRD5A1SRD5A2TUBB4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863898-A1 ENDOTHELIN RECEPTOR ANTAGONISTS MERCK PATENT GmbH (DE) 1998-09-16 EP disclosed
WO-1997019077-A1 ENDOTHELIN RECEPTOR ANTAGONISTS MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1997-05-29 WO disclosed