SCHEMBL8553723

SCHEMBL8553723

CCOC(=O)Oc1[nH]c2cc(OCc3ccccc3)ccc2c1-c1ccc(OC)cc1OCC(=O)O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 8/20 0.44
PPARD Q03181 7/20 0.42
PTPN1 P18031 2/20 0.42
FLT3 P36888 1/20 0.42
GABRA1 P14867 2/20 0.41
GABRG2 P18507 2/20 0.41
GABRB3 P28472 2/20 0.41
GABRA5 P31644 2/20 0.41
GABRA3 P34903 2/20 0.41
GABRA2 P47869 2/20 0.41
ALDH1A1 P00352 2/20 0.41
HPGD P15428 2/20 0.41
GABRP O00591 1/20 0.41
GABRD O14764 1/20 0.41
MAPT P10636 1/20 0.41
GABRB1 P18505 1/20 0.41
GABRB2 P47870 1/20 0.41
GABRA4 P48169 1/20 0.41
GABRE P78334 1/20 0.41
GABRA6 Q16445 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8550982 0.90 CTSV (0.44) FFAR1PPARDPTPN1GABRA1GABRG2
SCHEMBL8591475 0.85 PTPN1 (0.42) PTPN1GABRA1GABRG2GABRB3GABRA5
SCHEMBL8553299 0.80 PTPN1 (0.38) PTPN1GABRA1GABRG2GABRB3GABRA5
SCHEMBL8553319 0.78 PDE4B (0.40) PTPN1ALDH1A1HPGDMAPTMEN1
SCHEMBL8697633 0.77 POLB (0.37) PTPN1MEN1KMT2A
SCHEMBL8697275 0.77 PTPN1 (0.42) PTPN1ALDH1A1MAPTSMN1; SMN2
SCHEMBL8552298 0.74 EDNRA (0.53) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL8550354 0.74 ALDH1A1 (0.47) ALDH1A1HPGDMAPTMEN1KMT2A
SCHEMBL8551472 0.73 EDNRB (0.43) FFAR1PPARDPTPN1
SCHEMBL8551010 0.73 KDM4E (0.47) GABRA1GABRG2GABRB3GABRA5GABRA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863898-A1 ENDOTHELIN RECEPTOR ANTAGONISTS MERCK PATENT GmbH (DE) 1998-09-16 EP disclosed
WO-1997019077-A1 ENDOTHELIN RECEPTOR ANTAGONISTS MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1997-05-29 WO disclosed