SCHEMBL8552525

SCHEMBL8552525

CCCCCOc1cc2[nH]c(OC(=O)OCC)c(-c3ccc(OC)cc3OCC(=O)O)c2cc1OC

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ELANE P08246 3/20 0.38
SERPINE1 P05121 1/20 0.38
PTPN1 P18031 4/20 0.38
PLA2G4B P0C869 1/20 0.37
TSHR P16473 1/20 0.37
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
CYSLTR2 Q9NS75 1/20 0.36
CYSLTR1 Q9Y271 1/20 0.36
F2 P00734 2/20 0.36
MTNR1A P48039 1/20 0.35
MTNR1B P49286 1/20 0.35
KDM4E B2RXH2 3/20 0.35
ALDH1A1 P00352 3/20 0.35
HPGD P15428 3/20 0.35
MAPT P10636 3/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
GAA P10253 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8591475 0.93 PTPN1 (0.42) ELANEPTPN1KDM4EALDH1A1HPGD
SCHEMBL8550982 0.88 CTSV (0.44) ELANEPTPN1ALDH1A1HPGDMAPT
SCHEMBL8553299 0.88 PTPN1 (0.38) SERPINE1PTPN1KDM4EALDH1A1HPGD
SCHEMBL8553319 0.85 PDE4B (0.40) ELANEPTPN1KDM4EALDH1A1HPGD
SCHEMBL8553723 0.79 FFAR1 (0.44) PTPN1ALDH1A1HPGDMAPTMEN1
SCHEMBL8551010 0.78 KDM4E (0.47) ELANEKDM4EALDH1A1HPGDMAPT
SCHEMBL8549519 0.78 KDM4E (0.38) PDE3BPDE3AKDM4EALDH1A1HPGD
SCHEMBL8697275 0.74 PTPN1 (0.42) PTPN1ALDH1A1MAPTSMN1; SMN2
SCHEMBL8547163 0.73 EDNRB (0.45) ELANEPTPN1F2KDM4EGAA
SCHEMBL8546754 0.73 NPC1 (0.40) KDM4EALDH1A1HPGDMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863898-A1 ENDOTHELIN RECEPTOR ANTAGONISTS MERCK PATENT GmbH (DE) 1998-09-16 EP disclosed
WO-1997019077-A1 ENDOTHELIN RECEPTOR ANTAGONISTS MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1997-05-29 WO disclosed