SCHEMBL8551329

SCHEMBL8551329

NC(=O)COc1ccc2cc(OC[C@@H](O)CCc3cccnc3)ccc2c1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.45
MAPT P10636 2/20 0.45
LMNA P02545 1/20 0.45
HTT P42858 1/20 0.45
NAMPT P43490 1/20 0.43
F9 P00740 1/20 0.41
F10 P00742 1/20 0.41
ADRB1 P08588 1/20 0.40
ADRB3 P13945 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
POLB P06746 1/20 0.39
GPR132 Q9UNW8 2/20 0.39
MRGPRX4 Q96LA9 1/20 0.38
MAOB P27338 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8476796 1.00 ALDH1A1 (0.45) ALDH1A1MAPTLMNAHTTNAMPT
SCHEMBL8481177 0.87 SMN1; SMN2 (0.51) ALDH1A1MAPTLMNAHTTNAMPT
SCHEMBL8551036 0.87 SMN1; SMN2 (0.51) ALDH1A1MAPTLMNAHTTNAMPT
SCHEMBL8479757 0.86 POLB (0.52) ALDH1A1MAPTLMNAHTTNAMPT
SCHEMBL8479934 0.84 ADRB1 (0.45) ALDH1A1NAMPTF9F10ADRB1
SCHEMBL7964059 0.83 CYP3A4 (0.52) ALDH1A1MAPTLMNAHTTNAMPT
SCHEMBL8477139 0.83 ALOX5 (0.49) ALDH1A1LMNANAMPTF9F10
SCHEMBL7963443 0.83 CYP3A4 (0.52) ALDH1A1MAPTLMNAHTTNAMPT
SCHEMBL8480213 0.83 ALOX5 (0.49) ALDH1A1LMNANAMPTF9F10
SCHEMBL7771955 0.83 CA2 (0.44) NAMPTADRB1ADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0865431-A2 COMPOUNDS Astra Pharmaceuticals Limited (GB) 1998-09-23 EP disclosed
WO-1997020815-A1 COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1997-06-12 WO disclosed