SCHEMBL8551545

SCHEMBL8551545

O=C(COc1ccc(NC(=O)c2cnc(C3CCN(C(=O)OCc4ccccc4)CC3)s2)cc1)OC1CCCCC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 1/20 0.42
USP30 Q70CQ3 1/20 0.41
KDM4E B2RXH2 1/20 0.41
LMNA P02545 1/20 0.41
CXCR1 P25024 1/20 0.41
CXCR2 P25025 1/20 0.41
FLT3 P36888 1/20 0.41
GRIN2B Q13224 6/20 0.39
CYP2D6 P10635 3/20 0.39
CYP2C9 P11712 3/20 0.39
NPC1 O15118 3/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
CYP3A4 P08684 2/20 0.39
RAB9A P51151 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
MAPT P10636 2/20 0.39
ALDH1A1 P00352 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
PDE4B Q07343 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8551784 0.90 HTT (0.46) ENPP2USP30KDM4ELMNAFLT3
SCHEMBL8553111 0.77 SMN1; SMN2 (0.56) GRIN2BCYP2D6CYP2C9NPC1MEN1
SCHEMBL8551127 0.75 LMNA (0.45) ENPP2USP30KDM4ELMNAFLT3
SCHEMBL8626081 0.73 SMN1; SMN2 (0.51) GRIN2BCYP2D6CYP2C9NPC1MEN1
SCHEMBL8552625 0.72 LMNA (0.46) ENPP2LMNAGRIN2BMEN1KMT2A
SCHEMBL23201424 0.71 SMN1; SMN2 (0.57) GRIN2BCYP2D6CYP2C9NPC1MEN1
SCHEMBL8553852 0.71 HTT (0.45) ENPP2KDM4ELMNAGRIN2BCYP2D6
SCHEMBL2006749 0.70 SMN1; SMN2 (0.51) GRIN2BCYP2D6CYP2C9NPC1MEN1
Bromide SCHEMBL8551319 0.70 POLB (0.44) CXCR1CXCR2MEN1KMT2AALDH1A1
Hydrochloric Acid SCHEMBL8549386 0.70 POLB (0.48) KDM4ECXCR1CXCR2NPC1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0858457-A1 5-MEMBERED HETEROCYCLES, PHARMACEUTICAL AGENTS CONTAINING SAID COMPOUNDS AND THE USE THEREOF AND METHODS OF PRODUCING THEM Dr. Karl Thomae GmbH (DE) 1998-08-19 EP disclosed
WO-1997015567-A1 5-MEMBERED HETEROCYCLES, PHARMACEUTICAL AGENTS CONTAINING SAID COMPOUNDS AND THE USE THEREOF AND METHODS OF PRODUCING THEM DR. KARL THOMAE GMBH (DE) 1997-05-01 WO disclosed