SCHEMBL8553852

SCHEMBL8553852

COC(=O)CCN1CCC(NC(=O)c2cnc(C3CCN(C(=O)OCc4ccccc4)CC3)s2)CC1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.45
ENPP2 Q13822 3/20 0.44
SMN1; SMN2 Q16637 3/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
GRIN2B Q13224 4/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
TP53 P04637 1/20 0.41
LMNA P02545 1/20 0.41
THRB P10828 1/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
MAPK1 P28482 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8552625 0.80 LMNA (0.46) HTTENPP2GRIN2BMEN1KMT2A
Bromide SCHEMBL8593328 0.80 SMYD3 (0.38) SMN1; SMN2
SCHEMBL8553111 0.79 SMN1; SMN2 (0.56) HTTSMN1; SMN2NPC1RAB9AGRIN2B
SCHEMBL8551784 0.78 HTT (0.46) HTTENPP2SMN1; SMN2NPC1RAB9A
SCHEMBL8626081 0.77 SMN1; SMN2 (0.51) HTTSMN1; SMN2NPC1RAB9AGRIN2B
SCHEMBL8552781 0.74 LMNA (0.47) HTTENPP2SMN1; SMN2NPC1RAB9A
SCHEMBL23201424 0.73 SMN1; SMN2 (0.57) HTTSMN1; SMN2NPC1RAB9AGRIN2B
SCHEMBL2857988 0.73 HTT (0.62) HTTENPP2SMN1; SMN2NPC1RAB9A
SCHEMBL7137790 0.71 SMN1; SMN2 (0.65) HTTENPP2SMN1; SMN2NPC1RAB9A
SCHEMBL658800 0.70 LTA4H (0.59) MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0858457-A1 5-MEMBERED HETEROCYCLES, PHARMACEUTICAL AGENTS CONTAINING SAID COMPOUNDS AND THE USE THEREOF AND METHODS OF PRODUCING THEM Dr. Karl Thomae GmbH (DE) 1998-08-19 EP disclosed
WO-1997015567-A1 5-MEMBERED HETEROCYCLES, PHARMACEUTICAL AGENTS CONTAINING SAID COMPOUNDS AND THE USE THEREOF AND METHODS OF PRODUCING THEM DR. KARL THOMAE GMBH (DE) 1997-05-01 WO disclosed