SCHEMBL8552088

SCHEMBL8552088

CC(C)N1CCC(c2coc3ccc(NC(=O)Nc4cccc(Br)c4Br)cc23)CC1

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 12/20 0.39
HTR2A P28223 12/20 0.39
DRD3 P35462 12/20 0.39
MAPT P10636 2/20 0.38
TP53 P04637 1/20 0.38
ALDH1A1 P00352 2/20 0.37
EPHX2 P34913 2/20 0.35
RAB9A P51151 2/20 0.35
HTT P42858 1/20 0.35
ATAD2 Q6PL18 1/20 0.34
CECR2 Q9BXF3 1/20 0.34
NPC1 O15118 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8548045 0.90 DRD2 (0.34) DRD2HTR2ADRD3ALDH1A1HTT
SCHEMBL8704542 0.85 ALDH1A1 (0.53) DRD2HTR2ADRD3ALDH1A1EPHX2
SCHEMBL8548755 0.84 CA2 (0.43) DRD2HTR2ADRD3MAPTTP53
SCHEMBL7483808 0.82 HTR1D (0.55) DRD2
SCHEMBL8549413 0.81 ALDH1A1 (0.40) DRD2HTR2ADRD3MAPTTP53
Hydrochloric Acid SCHEMBL8549247 0.75 TP53 (0.46) DRD2HTR2ADRD3MAPTTP53
SCHEMBL8547778 0.75 DRD2 (0.41) DRD2HTR2ADRD3MAPTRAB9A
SCHEMBL8548758 0.75 DRD2 (0.40) DRD2HTR2ADRD3TP53ALDH1A1
SCHEMBL8552340 0.73 DRD2 (0.47) DRD2HTR2ADRD3MAPT
SCHEMBL8546763 0.73 HTR1D (0.45) DRD2HTR2ADRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5792763-A MIGRAINES; ANALGESICS; DISEASES LINKED TO DECREASED NEUROTRANMISSION OF SEROTONIN IN MAMMALS ELI LILLY AND COMPANY (US) 1998-08-11 US disclosed
EP-0835869-A2 New serotonin 5-HT1F agonists ELI LILLY AND COMPANY (US) 1998-04-15 EP disclosed