SCHEMBL8552154

SCHEMBL8552154

Clc1nnc(-c2ccccc2)c2occc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.38
PKM P14618 1/20 0.38
ADORA2A P29274 5/20 0.36
ADORA1 P30542 5/20 0.36
LMNA P02545 6/20 0.35
SMN1; SMN2 Q16637 4/20 0.35
HTT P42858 3/20 0.35
ALDH1A1 P00352 3/20 0.35
L3MBTL1 Q9Y468 3/20 0.35
MAPK1 P28482 2/20 0.35
KMT2A Q03164 2/20 0.35
GLA P06280 1/20 0.35
HPGD P15428 1/20 0.35
MEN1 O00255 1/20 0.35
TP53 P04637 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
MAPT P10636 2/20 0.35
NPSR1 Q6W5P4 2/20 0.35
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL580485 0.86 LMNA (0.38) KDM4EPKMADORA2AADORA1LMNA
SCHEMBL3606506 0.77 GOT1 (0.32)
SCHEMBL580414 0.74 MAPT (0.49) KDM4EPKMLMNASMN1; SMN2HTT
SCHEMBL29537275 0.74 MAPT (0.49) KDM4EPKMLMNASMN1; SMN2HTT
SCHEMBL581638 0.72 LMNA (0.37) KDM4EADORA2AADORA1LMNAHTT
SCHEMBL8551380 0.69 LMNA (0.45) KDM4EPKMADORA2AADORA1LMNA
SCHEMBL28471578 0.68 KDM4E (0.44) KDM4EPKMADORA2AADORA1LMNA
SCHEMBL7262166 0.68 MAOA (0.45) KDM4EPKMADORA2ASMN1; SMN2ALDH1A1
SCHEMBL9138181 0.67 KDM4E (0.47) KDM4EPKMADORA2AADORA1LMNA
SCHEMBL1316871 0.67 PTGS1 (0.41) KDM4EPKMLMNASMN1; SMN2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0534443-B1 3,6-Disubstituted pyridazine derivatives MITSUBISHI CHEM CORP (JP) 1998-12-30 EP disclosed
US-5462941-A 1-(cyclohexylalkylamino)-4-(phenyl, thienyl, or furyl) phthalazines; anti-platelet agglutination agents for treatment or prevention of cerebro- or cardiovascular disorders MITSUBISHI CHEMICAL CORPORATION (JP) 1995-10-31 US disclosed
EP-0534443-A1 3,6-Disubstituted pyridazine derivatives Mitsubishi Chemical Corporation (JP) 1993-03-31 EP disclosed