SCHEMBL8552273

SCHEMBL8552273

COC(=O)C(Cc1ccoc1)N1C(=O)CC1SCc1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ACE P12821 1/20 0.37
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
CHRM2 P08172 1/20 0.35
CHRM1 P11229 1/20 0.35
CHRM3 P20309 1/20 0.35
ALDH1A1 P00352 1/20 0.34
PKM P14618 1/20 0.34
GAA P10253 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8552490 0.90 ALDH1A1 (0.42) ACENPC1RAB9AALDH1A1PKM
SCHEMBL8552104 0.89 ALDH1A1 (0.42) ACEALDH1A1PKMGAA
SCHEMBL8557349 0.83 L3MBTL1 (0.40) ACENPC1RAB9AALDH1A1
SCHEMBL8550015 0.81 ACE (0.38) ACEALDH1A1GAA
SCHEMBL8557133 0.79 ACE (0.37) ACEALDH1A1
SCHEMBL8551020 0.78 ACE (0.43) ACEALDH1A1
SCHEMBL8554773 0.77 ALDH1A1 (0.54) ACEALDH1A1PKMGAA
SCHEMBL8556164 0.77 HDAC3 (0.39) NPC1RAB9A
SCHEMBL5170081 0.74 GAA (0.42) ACENPC1RAB9AALDH1A1GAA
SCHEMBL27484036 0.74 ACE (0.40) ACEALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0840725-A1 AZETIDINONE DERIVATIVES FOR THE TREATMENT OF ATHEROSCLEROSIS SMITHKLINE BEECHAM PLC (GB) 1998-05-13 EP disclosed
WO-1997002242-A1 AZETIDINONE DERIVATIVES FOR THE TREATMENT OF ATHEROSCLEROSIS SMITHKLINE BEECHAM PLC (GB) 1997-01-23 WO disclosed