SCHEMBL8552464

SCHEMBL8552464

Cc1ccccc1-c1nnc(Cl)c2c(Br)cccc12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.37
HSD11B1 P28845 1/20 0.37
ALDH1A1 P00352 2/20 0.36
SMO Q99835 1/20 0.36
CYP1A2 P05177 2/20 0.35
NPC1 O15118 5/20 0.34
RAB9A P51151 5/20 0.34
SMN1; SMN2 Q16637 4/20 0.34
CASP3 P42574 1/20 0.34
SENP8 Q96LD8 1/20 0.34
SENP7 Q9BQF6 1/20 0.34
SENP6 Q9GZR1 1/20 0.34
HPGD P15428 2/20 0.34
MAOB P27338 2/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
MAPT P10636 2/20 0.34
KDM4E B2RXH2 1/20 0.34
APAF1 O14727 1/20 0.34
TDP2 O95551 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8547106 0.88 SMO (0.41) ADORA2AALDH1A1SMOCYP1A2NPC1
SCHEMBL8549331 0.85 HSD11B1 (0.42) HSD11B1ALDH1A1SMOCYP1A2NPC1
SCHEMBL8550501 0.82 HSD11B1 (0.34) HSD11B1ALDH1A1AR
SCHEMBL8552471 0.82 ADORA2A (0.40) ADORA2AALDH1A1SMOCYP1A2NPC1
SCHEMBL8546655 0.82 MAPK1 (0.42) HSD11B1ALDH1A1CYP1A2NPC1RAB9A
SCHEMBL8547547 0.79 SMO (0.44) ADORA2AALDH1A1SMONPC1RAB9A
SCHEMBL8548393 0.79 HSD11B1 (0.44) HSD11B1KDR
SCHEMBL8549262 0.78 ALDH1A1 (0.41) ADORA2AALDH1A1CYP1A2SMN1; SMN2HPGD
SCHEMBL8372792 0.76 PLAU (0.43) ADORA2AALDH1A1SMOCYP1A2HPGD
Hydrochloric Acid SCHEMBL8551595 0.75 PLAU (0.42) ADORA2AALDH1A1SMOCYP1A2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825187-A1 Condensed pyridazinyl guanidines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-25 EP disclosed