SCHEMBL8549331

SCHEMBL8549331

Clc1ccccc1-c1nnc(Cl)c2c(Br)cccc12

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 2/20 0.42
SMN1; SMN2 Q16637 3/20 0.38
SMO Q99835 1/20 0.37
CYP1A2 P05177 1/20 0.36
ELANE P08246 1/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
TP53 P04637 1/20 0.36
HPGD P15428 1/20 0.36
GPR84 Q9NQS5 1/20 0.36
MAOB P27338 1/20 0.36
KMT2A Q03164 2/20 0.35
GAA P10253 1/20 0.35
PTGES O14684 2/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
RXFP1 Q9HBX9 1/20 0.33
CRHR1 P34998 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8546655 0.85 MAPK1 (0.42) HSD11B1SMN1; SMN2CYP1A2NPC1RAB9A
SCHEMBL8552464 0.85 ADORA2A (0.37) HSD11B1SMN1; SMN2SMOCYP1A2ELANE
SCHEMBL8548393 0.81 HSD11B1 (0.44) HSD11B1
SCHEMBL8549262 0.81 ALDH1A1 (0.41) SMN1; SMN2CYP1A2HPGDKMT2AALDH1A1
SCHEMBL8549276 0.78 PLAU (0.43) HSD11B1SMN1; SMN2SMOKMT2AGAA
SCHEMBL8549269 0.76 HSD11B1 (0.34) HSD11B1SMN1; SMN2SMOGPR84MAOB
SCHEMBL8551565 0.76 KMT2A (0.42) SMN1; SMN2SMOCYP1A2NPC1RAB9A
SCHEMBL8551877 0.74 ESR1 (0.37) SMN1; SMN2SMOCYP1A2HPGDGPR84
SCHEMBL8552195 0.74 AR (0.42) HSD11B1SMN1; SMN2CYP1A2ELANENPC1
SCHEMBL28934596 0.72 L3MBTL1 (0.37) SMN1; SMN2CYP1A2NPC1RAB9AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825187-A1 Condensed pyridazinyl guanidines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-25 EP disclosed