SCHEMBL8550501

SCHEMBL8550501

Cc1cc(F)ccc1-c1nnc(Cl)c2c(Br)cccc12

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 2/20 0.34
MAPK14 Q16539 7/20 0.33
HSP90AB1 P08238 5/20 0.32
GRM2 Q14416 1/20 0.32
PARP1 P09874 1/20 0.31
AR P10275 1/20 0.30
P2RX7 Q99572 1/20 0.30
RXFP1 Q9HBX9 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8552464 0.82 ADORA2A (0.37) HSD11B1ARALDH1A1
SCHEMBL8372826 0.79 PLAU (0.39) MAPK14ALDH1A1
SCHEMBL8551877 0.78 ESR1 (0.37) MAPK14GRM2ALDH1A1
Hydrochloric Acid SCHEMBL8552094 0.78 PLAU (0.38) MAPK14ALDH1A1
SCHEMBL8372825 0.77 ENPP3 (0.33) MAPK14HSP90AB1ALDH1A1
SCHEMBL8546629 0.75 PARP1 (0.40) PARP1
SCHEMBL28934596 0.75 L3MBTL1 (0.37) HSP90AB1ALDH1A1
SCHEMBL8549331 0.74 HSD11B1 (0.42) HSD11B1RXFP1ALDH1A1
SCHEMBL8548393 0.71 HSD11B1 (0.44) HSD11B1
SCHEMBL8549262 0.70 ALDH1A1 (0.41) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825187-A1 Condensed pyridazinyl guanidines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-25 EP disclosed