SCHEMBL8552785

SCHEMBL8552785

CCN(CCOC(=O)C(C)(C)C)CCOc1ccc2nc(Cc3ccc(F)cc3)sc2c1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.49
CYP1A2 P05177 1/20 0.48
CYP2D6 P10635 1/20 0.48
CACNA1B Q00975 3/20 0.43
MAPT P10636 1/20 0.41
HTT P42858 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
HDAC6 Q9UBN7 1/20 0.39
CA1 P00915 7/20 0.38
CA2 P00918 7/20 0.38
CA4 P22748 2/20 0.38
PPARD Q03181 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8554328 0.92 LMNA (0.48) LMNACYP1A2CYP2D6CACNA1BMAPT
SCHEMBL8361641 0.91 LMNA (0.49) LMNACYP1A2CYP2D6MAPTHTT
SCHEMBL8359973 0.87 LMNA (0.60) LMNACYP1A2CYP2D6CACNA1BMAPT
SCHEMBL8552900 0.86 LMNA (0.53) LMNACYP1A2CYP2D6CACNA1BMAPT
SCHEMBL8359946 0.82 THRB (0.42) LMNAL3MBTL1HDAC6
SCHEMBL8357762 0.81 LMNA (0.49) LMNACYP1A2CYP2D6MAPTHTT
SCHEMBL8357917 0.79 HTT (0.48) LMNACYP1A2CYP2D6CACNA1BMAPT
SCHEMBL8551252 0.79 LMNA (0.50) LMNACYP1A2CYP2D6CACNA1BMAPT
SCHEMBL8356218 0.77 LMNA (0.60) LMNACYP1A2CYP2D6HTT
SCHEMBL8361490 0.77 LMNA (0.53) LMNACYP1A2CYP2D6MAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0824529-A1 BENZOTHIAZOLES AND BENZOXAZOLES, AS WELL AS DRUGS CONTAINING THEM, THEIR USE AND METHODS OF PREPARING THEM Dr. Karl Thomae GmbH (DE) 1998-02-25 EP disclosed
WO-1996035681-A1 BENZOTHIAZOLES AND BENZOXAZOLES, AS WELL AS DRUGS CONTAINING THEM, THEIR USE AND METHODS OF PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-11-14 WO disclosed