SCHEMBL8552914

SCHEMBL8552914

CC(=O)Nc1cccc(-c2ccc(OC(CC(C)O)c3cccnc3)cc2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 9/20 0.48
CYP11B1 P15538 2/20 0.48
CYP11B2 P19099 2/20 0.48
ITGB3 P05106 1/20 0.46
ITGAV P06756 1/20 0.46
ITGA2B P08514 1/20 0.46
FYN P06241 2/20 0.45
CYP3A4 P08684 2/20 0.44
PIP4K2A P48426 1/20 0.43
PIP4K2B P78356 1/20 0.43
PTGIR P43119 2/20 0.42
LMNA P02545 1/20 0.41
POLB P06746 1/20 0.41
PKM P14618 1/20 0.41
KMT2A Q03164 1/20 0.41
PSEN1 P49768 1/20 0.41
PSEN2 P49810 1/20 0.41
APH1B Q8WW43 1/20 0.41
NCSTN Q92542 1/20 0.41
APH1A Q96BI3 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8555638 0.87 SUCNR1 (0.43) FYNLMNAKMT2A
SCHEMBL8118375 0.86 KCNA5 (0.49) FYNCYP3A4PIP4K2APIP4K2B
SCHEMBL8554677 0.84 EPHX1 (0.42) LMNAPKM
SCHEMBL8551743 0.83 KMO (0.51) LMNA
SCHEMBL8552459 0.83 CYP17A1 (0.44) CYP17A1CYP11B1CYP11B2CYP3A4
SCHEMBL8552624 0.82 CYP19A1 (0.47) CYP17A1CYP11B1CYP11B2CYP3A4
SCHEMBL8109544 0.82 SMN1; SMN2 (0.44) CYP17A1CYP3A4PKM
SCHEMBL8118468 0.82 KCNA5 (0.45) CYP17A1CYP11B1CYP11B2CYP3A4
SCHEMBL8118689 0.82 KCNA5 (0.48) CYP17A1CYP11B1CYP11B2CYP3A4
SCHEMBL8118264 0.82 DGAT2 (0.39) CYP17A1CYP11B1CYP11B2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0865431-A2 COMPOUNDS Astra Pharmaceuticals Limited (GB) 1998-09-23 EP disclosed
WO-1997020815-A1 COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1997-06-12 WO disclosed