SCHEMBL8552963

SCHEMBL8552963

N=C(N)Nc1nnc(-c2ccccn2)c2cc(Cl)c(Cl)cc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.39
ADORA1 P30542 2/20 0.39
ADORA3 P0DMS8 4/20 0.34
GABRA1 P14867 1/20 0.34
TACR2 P21452 1/20 0.34
OPRD1 P41143 1/20 0.34
KMT5B Q4FZB7 1/20 0.34
KMT5C Q86Y97 1/20 0.34
NPC1 O15118 1/20 0.34
MAPT P10636 1/20 0.34
RAB9A P51151 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
CCR1 P32246 1/20 0.34
CCR5 P51681 1/20 0.34
CCR8 P51685 1/20 0.34
GRM4 Q14833 1/20 0.34
NPY5R Q15761 1/20 0.34
SLC2A1 P11166 1/20 0.34
PIK3CD O00329 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8547080 0.82 KDR (0.43) ADORA2AADORA1ADORA3GABRA1TACR2
SCHEMBL8552965 0.75 PLAU (0.44) ADORA2AADORA1ADORA3NPSR1RXFP1
SCHEMBL8552255 0.75 ADORA2A (0.44) ADORA2AADORA1NPC1MAPTRAB9A
SCHEMBL8548292 0.74 ADORA2A (0.41) ADORA2AADORA1ADORA3GABRA1TACR2
SCHEMBL8553138 0.71 POLB (0.37) NPC1MAPTRAB9ANPSR1RXFP1
SCHEMBL8551930 0.65 NPSR1 (0.51) MAPTNPSR1
Hydrochloric Acid SCHEMBL8550943 0.64 NPSR1 (0.50) MAPTNPSR1
SCHEMBL9807627 0.64 METAP1 (0.47) ADORA2AADORA1NPC1MAPTRAB9A
Hydrochloric Acid SCHEMBL8548606 0.63 ALDH1A1 (0.42) MAPTNPSR1
SCHEMBL8549645 0.62 LRRK2 (0.53) NPC1RAB9ANPSR1CCR1CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825187-A1 Condensed pyridazinyl guanidines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-25 EP disclosed