SCHEMBL8553138

SCHEMBL8553138

N=C(N)Nc1nnc(-c2ccccn2)c2cccc([N+](=O)[O-])c12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.37
NPC1 O15118 5/20 0.37
F12 P00748 1/20 0.36
ALDH1A1 P00352 3/20 0.35
NSUN3 Q9H649 1/20 0.35
KMT2A Q03164 4/20 0.35
MEN1 O00255 3/20 0.35
CTSB P07858 2/20 0.35
GAA P10253 2/20 0.35
MAPT P10636 2/20 0.35
KDM4E B2RXH2 1/20 0.35
IDO1 P14902 1/20 0.35
TDO2 P48775 1/20 0.35
NCOA1 Q15788 1/20 0.35
NCOA3 Q9Y6Q9 1/20 0.35
ABCG2 Q9UNQ0 1/20 0.35
NPSR1 Q6W5P4 2/20 0.34
S1PR4 O95977 1/20 0.34
HPGD P15428 1/20 0.34
XBP1 P17861 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8550910 0.84 ABCG2 (0.39) ALDH1A1KMT2AMEN1MAPTKDM4E
SCHEMBL8552276 0.80 KDR (0.43) POLBNPC1ALDH1A1KMT2AMEN1
SCHEMBL8553148 0.78 PLAU (0.42) POLBNPC1F12ALDH1A1KMT2A
SCHEMBL8551326 0.77 ALDH1A1 (0.44) POLBNPC1ALDH1A1KMT2AMEN1
SCHEMBL8552963 0.71 ADORA2A (0.39) NPC1MAPTNPSR1RAB9ARXFP1
SCHEMBL8548686 0.69 LRRK2 (0.49) POLBNPC1ALDH1A1KMT2AMEN1
SCHEMBL16387910 0.66 PDE10A (0.50) POLBNPC1F12ALDH1A1KMT2A
Hydrochloric Acid SCHEMBL8546714 0.66 MEN1 (0.45) NPC1ALDH1A1KMT2AMEN1GAA
SCHEMBL4150422 0.66 PDE10A (0.53) POLBNPC1F12ALDH1A1KMT2A
SCHEMBL30117516 0.66 PDE10A (0.53) POLBNPC1F12ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825187-A1 Condensed pyridazinyl guanidines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-25 EP disclosed