SCHEMBL8552965

SCHEMBL8552965

NC(N)=Nc1nnc(-c2ccccn2)c2cc(Cl)c(Cl)cc12

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PLAU P00749 11/20 0.44
SLC2A1 P11166 1/20 0.43
ADORA3 P0DMS8 1/20 0.42
PLG P00747 2/20 0.42
HSP90AA1 P07900 1/20 0.41
ADORA2A P29274 1/20 0.41
ADORA1 P30542 1/20 0.41
ADRA2A P08913 2/20 0.41
ADRA2B P18089 2/20 0.41
ADRA2C P18825 2/20 0.41
F9 P00740 1/20 0.38
CCR1 P32246 1/20 0.36
CCR5 P51681 1/20 0.36
CCR8 P51685 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8547084 0.80 PLAU (0.51) PLAUPLGADORA2AADORA1F9
SCHEMBL8552255 0.78 ADORA2A (0.44) HSP90AA1ADORA2AADORA1CCR1CCR5
SCHEMBL8552963 0.75 ADORA2A (0.39) SLC2A1ADORA3ADORA2AADORA1CCR1
SCHEMBL8548298 0.72 PLAU (0.40) PLAUADORA3PLGADORA2AADORA1
SCHEMBL8553148 0.71 PLAU (0.42) PLAUSLC2A1ADORA3PLGHSP90AA1
SCHEMBL9807627 0.66 METAP1 (0.47) HSP90AA1ADORA2AADORA1CCR1CCR5
SCHEMBL8549645 0.65 LRRK2 (0.53) CCR1CCR5CCR8NPSR1
SCHEMBL7952022 0.65 KDM4E (0.70) HSP90AA1ADORA2AADORA1CCR1CCR5
SCHEMBL8551931 0.64 PLG (0.53) PLAUPLGNPSR1
SCHEMBL9775492 0.63 KDM4E (0.56) HSP90AA1ADORA2AADORA1CCR1CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825187-A1 Condensed pyridazinyl guanidines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-25 EP disclosed