SCHEMBL8553148

SCHEMBL8553148

NC(N)=Nc1nnc(-c2ccccn2)c2cccc([N+](=O)[O-])c12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLAU P00749 4/20 0.42
NPC1 O15118 4/20 0.39
RAB9A P51151 3/20 0.39
POLB P06746 2/20 0.39
PLG P00747 2/20 0.39
MAPK1 P28482 1/20 0.39
F12 P00748 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
NCOA1 Q15788 1/20 0.36
NCOA3 Q9Y6Q9 1/20 0.36
HSP90AA1 P07900 1/20 0.36
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
S1PR4 O95977 1/20 0.35
HPGD P15428 1/20 0.35
XBP1 P17861 1/20 0.35
S1PR1 P21453 1/20 0.35
CCR6 P51684 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
ALDH1A1 P00352 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8550917 0.83 PLAU (0.45) PLAUNPC1RAB9APLGMAPK1
SCHEMBL8551326 0.79 ALDH1A1 (0.44) NPC1RAB9APOLBNCOA1NCOA3
SCHEMBL8552284 0.79 PLAU (0.40) PLAUNPC1RAB9APOLBPLG
SCHEMBL8553138 0.78 POLB (0.37) NPC1RAB9APOLBMAPK1F12
SCHEMBL8552965 0.71 PLAU (0.44) PLAUPLGADORA3HSP90AA1NPSR1
SCHEMBL8548686 0.71 LRRK2 (0.49) NPC1RAB9APOLBMAPK1NCOA1
SCHEMBL16387910 0.68 PDE10A (0.50) NPC1RAB9APOLBF12NCOA1
SCHEMBL4150422 0.67 PDE10A (0.53) NPC1RAB9APOLBMAPK1F12
SCHEMBL30117516 0.67 PDE10A (0.53) NPC1RAB9APOLBMAPK1F12
SCHEMBL11224715 0.66 F12 (0.52) NPC1RAB9AMAPK1F12MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825187-A1 Condensed pyridazinyl guanidines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-25 EP disclosed