SCHEMBL8553475

SCHEMBL8553475

CCc1ccc(-c2nc(CN3CCN(CC(=O)Nc4c(C)cccc4C)CC3)oc2-c2ccc(CC)cc2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.45
DRD4 P21917 2/20 0.41
TP53 P04637 1/20 0.41
REV1 Q9UBZ9 1/20 0.41
ALDH1A1 P00352 3/20 0.41
ADRB1 P08588 2/20 0.40
CYP3A4 P08684 2/20 0.40
ADRA2A P08913 2/20 0.40
CYP2D6 P10635 2/20 0.40
ADRA2B P18089 2/20 0.40
ADRA2C P18825 2/20 0.40
ADRA1A P35348 2/20 0.40
DRD3 P35462 2/20 0.40
HTR2B P41595 2/20 0.40
KCNH2 Q12809 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
MLNR O43193 1/20 0.40
NR1I2 O75469 1/20 0.40
USP2 O75604 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8554703 0.98 GAA (0.43) GAADRD4TP53REV1ALDH1A1
SCHEMBL8552887 0.91 NR4A2 (0.47) ALDH1A1ADRB1CYP3A4ADRA2ACYP2D6
SCHEMBL8557576 0.90 MEN1 (0.52) GAADRD4REV1ALDH1A1ADRB1
SCHEMBL8557330 0.87 CETP (0.43) GAAALDH1A1ADRB1CYP3A4ADRA2A
SCHEMBL8552938 0.83 RXRA (0.46) GAADRD4ALDH1A1KCNH2KMT2A
SCHEMBL8555057 0.81 NR4A2 (0.51) DRD4ADRB1CYP3A4ADRA2ACYP2D6
SCHEMBL8554568 0.79 KDR (0.58) GAAALDH1A1CYP3A4ADRA1ADRD3
SCHEMBL8558360 0.79 RXRA (0.50) ADRB1CYP3A4ADRA2ACYP2D6ADRA2B
Hydrochloric Acid SCHEMBL8552139 0.78 CACNA1G (0.49) GAADRD4TP53REV1ALDH1A1
SCHEMBL8554363 0.78 KDR (0.57) TP53MEN1KMT2ALMNARXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0582164-B1 Adenosine re-uptake inhibiting derivatives of diphenyl oxazoles, thiazoles and imidazoles BRISTOL MYERS SQUIBB CO (US) 1998-12-23 EP claimed
US-5382584-A Antiischemic agents BRISTOL-MYERS SQUIBB COMPANY (US) 1995-01-17 US claimed
EP-0582164-A1 Adenosine re-uptake inhibiting derivatives of diphenyl oxazoles, thiazoles and imidazoles Bristol-Myers Squibb Company (US) 1994-02-09 EP claimed