SCHEMBL8553781

SCHEMBL8553781

O=C1CC(Oc2ccc(Cl)cc2)N1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 5/20 0.43
SLC6A2 P23975 4/20 0.43
SLC6A3 Q01959 4/20 0.43
MMP13 P45452 1/20 0.36
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34
SOD1 P00441 1/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
ALOX5 P09917 1/20 0.34
LSS P48449 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8552429 0.81 GAA (0.45) MEN1KMT2ACA1CA2CA9
SCHEMBL7360048 0.80 ALOX5 (0.50) SLC6A4SLC6A2SLC6A3ALOX5
SCHEMBL8814238 0.77 SMN1; SMN2 (0.37) MEN1KMT2AALDH1A1LMNANPC1
SCHEMBL6535358 0.76 SLC6A4 (0.50) SLC6A4SLC6A2SLC6A3
SCHEMBL8442229 0.74 SLC6A3 (0.43) SLC6A4SLC6A2SLC6A3MEN1KMT2A
SCHEMBL4789557 0.66 SLC6A4 (0.44) SLC6A4SLC6A2SLC6A3
SCHEMBL232806 0.65 SLC6A4 (0.63) SLC6A4SLC6A2SLC6A3
SCHEMBL11874603 0.65 MMP13 (0.47) SLC6A4SLC6A2SLC6A3MMP13MEN1
SCHEMBL5520546 0.65 SLC6A4 (0.51) SLC6A4SLC6A2SLC6A3MMP13MEN1
SCHEMBL1499046 0.64 TP53 (0.41) SLC6A4SLC6A2SLC6A3MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0840725-A1 AZETIDINONE DERIVATIVES FOR THE TREATMENT OF ATHEROSCLEROSIS SMITHKLINE BEECHAM PLC (GB) 1998-05-13 EP disclosed
WO-1997002242-A1 AZETIDINONE DERIVATIVES FOR THE TREATMENT OF ATHEROSCLEROSIS SMITHKLINE BEECHAM PLC (GB) 1997-01-23 WO disclosed