SCHEMBL8554476

SCHEMBL8554476

N=C(N)NCCc1ccc(OCCC2Oc3ccccc3N(Cc3ccc(C(=O)O)cc3)C2=O)cc1

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.46
ALDH1A1 P00352 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
TP53 P04637 1/20 0.41
PTPN1 P18031 2/20 0.40
PTPN2 P17706 1/20 0.40
ACP1 P24666 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
PPARG P37231 11/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8595844 0.92 TSHR (0.45) TSHRALDH1A1SMN1; SMN2TP53PPARG
SCHEMBL8604494 0.90 ALDH1A1 (0.43) TSHRALDH1A1SMN1; SMN2TP53PPARG
SCHEMBL8557727 0.90 GSK3B (0.47) TSHRALDH1A1SMN1; SMN2TP53PTPN1
SCHEMBL7475653 0.89 ALDH1A1 (0.42) TSHRALDH1A1SMN1; SMN2TP53PPARG
SCHEMBL8604038 0.88 TP53 (0.42) TSHRALDH1A1SMN1; SMN2TP53PPARG
SCHEMBL8554310 0.87 TSHR (0.48) TSHRALDH1A1SMN1; SMN2PTPN1PTPN2
SCHEMBL8556736 0.87 SIRT2 (0.41) TSHRALDH1A1SMN1; SMN2TP53MEN1
SCHEMBL8603405 0.87 TSHR (0.42) TSHRALDH1A1SMN1; SMN2TP53MEN1
SCHEMBL7476790 0.87 TSHR (0.45) TSHRALDH1A1SMN1; SMN2TP53PPARG
SCHEMBL8604319 0.86 ALDH1A1 (0.40) TSHRALDH1A1SMN1; SMN2TP53PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0869949-A1 BENZOXAZINE ANTIMICROBIAL AGENTS ORTHO PHARMACEUTICAL CORPORATION (US) 1998-10-14 EP disclosed
WO-1997017333-A1 BENZOXAZINE ANTIMICROBIAL AGENTS ORTHO PHARMACEUTICAL CORPORATION (US) 1997-05-15 WO disclosed