SCHEMBL8554951

SCHEMBL8554951

COc1ccc(N2CCN(C(CNC(=O)c3ccc4c(c3)CCOC4)(C(=O)OC(C)(C)C)C(=O)OC(C)(C)C)CC2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.47
MAPT P10636 2/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
ALDH1A1 P00352 2/20 0.45
GFER P55789 1/20 0.45
KDM4E B2RXH2 1/20 0.45
DRD2 P14416 5/20 0.43
HTR1D P28221 5/20 0.43
HTR2A P28223 5/20 0.43
DRD4 P21917 3/20 0.43
HTR1A P08908 3/20 0.43
HTR1B P28222 1/20 0.43
KMT2A Q03164 2/20 0.41
DRD3 P35462 1/20 0.40
MEN1 O00255 1/20 0.40
POLB P06746 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
OPRM1 P35372 1/20 0.39
OPRD1 P41143 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8550899 0.84 LMNA (0.37) LMNAMAPTSMN1; SMN2ALDH1A1DRD2
SCHEMBL8551589 0.80 USP5 (0.39) LMNASMN1; SMN2ALDH1A1KDM4EDRD2
SCHEMBL8549853 0.80 DRD4 (0.65) MAPTSMN1; SMN2ALDH1A1DRD2HTR1D
SCHEMBL8549327 0.74 DRD2 (0.39) LMNAMAPTSMN1; SMN2ALDH1A1GFER
SCHEMBL8549609 0.70 DRD4 (0.58) DRD2HTR1DHTR2ADRD4HTR1A
SCHEMBL8550144 0.69 DRD2 (0.50) DRD2HTR1DHTR2ADRD4HTR1A
SCHEMBL8548777 0.69 HTR1D (0.54) DRD2HTR1DHTR2ADRD4HTR1A
SCHEMBL8550575 0.68 DRD2 (0.49) DRD2HTR1DHTR2ADRD4HTR1A
SCHEMBL8553219 0.68 HTR1A (0.52) MAPTDRD2DRD4HTR1ADRD3
SCHEMBL8550457 0.68 HTR1A (0.51) MAPTDRD2DRD4HTR1ADRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0836599-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1998-04-22 EP disclosed