SCHEMBL8554964

SCHEMBL8554964

NC1N=C(CN2CCOCC2)c2ccccc2N(CC(=O)N2CCCC2)C1=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.48
KMT2A Q03164 5/20 0.43
MEN1 O00255 4/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
CCKBR P32239 4/20 0.42
KDM4E B2RXH2 4/20 0.41
GAA P10253 3/20 0.41
HSD17B10 Q99714 1/20 0.40
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
ALDH3A1 P30838 1/20 0.39
HTT P42858 1/20 0.39
TP53 P04637 1/20 0.39
MAPT P10636 1/20 0.39
THRB P10828 1/20 0.39
ALOX12 P18054 1/20 0.39
MAPK1 P28482 1/20 0.39
ATM Q13315 1/20 0.39
POLB P06746 1/20 0.38
HPGD P15428 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8553824 0.81 POLB (0.41) ALDH1A1KMT2AMEN1CA1CA2
SCHEMBL8558106 0.80 SENP1 (0.49) ALDH1A1CCKBR
SCHEMBL8555947 0.78 HRH3 (0.38) ALDH1A1SMN1; SMN2KDM4ECA1CA2
SCHEMBL9865548 0.78 CCKBR (0.61) ALDH1A1CCKBRHSD17B10TP53
SCHEMBL9573427 0.78 CCKBR (0.61) ALDH1A1CCKBRHSD17B10TP53
Bromide SCHEMBL9592670 0.77 CCKBR (0.61) ALDH1A1CCKBRHSD17B10TP53
Bromide SCHEMBL9592675 0.77 CCKBR (0.61) ALDH1A1CCKBRHSD17B10TP53
SCHEMBL9573650 0.76 ALDH1A1 (0.52) ALDH1A1KMT2AMEN1CCKBRHSD17B10
SCHEMBL9007296 0.73 CCKBR (0.55) CCKBR
SCHEMBL1388537 0.73 CCKBR (0.55) CCKBR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0672037-B1 1,4-BENZODIAZEPINE DERIVATIVES AND THEIR USE AS CCK-MODULATORS GLAXO GROUP LTD (GB) 1998-07-08 EP disclosed
US-5569654-A ADMINISTERING AS ANTAGONISTS OF GASTRIN AND CHOLECYSTOKININ GLAXO GROUP LIMITED (GB) 1996-10-29 US disclosed