SCHEMBL8555947

SCHEMBL8555947

CCN(C(=O)CN1C(=O)C(N)N=C(CN2CCOCC2)c2ccccc21)c1ccc(F)cc1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.38
POLB P06746 2/20 0.37
ALDH1A1 P00352 5/20 0.35
KDM4E B2RXH2 1/20 0.35
TSHR P16473 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.34
ALDH3A1 P30838 2/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
ACHE P22303 1/20 0.34
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34
HIF1A Q16665 1/20 0.34
KCNH2 Q12809 1/20 0.34
UBE2M P61081 1/20 0.34
DCUN1D1 Q96GG9 1/20 0.34
OXTR P30559 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1388570 0.85 CCKBR (0.49)
SCHEMBL8553824 0.84 POLB (0.41) HRH3POLBALDH1A1ALDH3A1CA1
SCHEMBL8555082 0.83 SENP1 (0.44) OXTR
SCHEMBL8554964 0.78 ALDH1A1 (0.48) POLBALDH1A1KDM4EALDH3A1CA1
SCHEMBL9573630 0.73 GABRP (0.54) POLBALDH1A1OXTR
SCHEMBL8554771 0.72 CCKBR (0.49)
SCHEMBL8555248 0.72 OXTR (0.41) POLBOXTR
SCHEMBL8555289 0.71 CCKBR (0.45) OXTR
SCHEMBL9007294 0.71 CCKBR (0.46)
SCHEMBL9007270 0.69 CCKBR (0.39) POLBALDH1A1HIF1ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0672037-B1 1,4-BENZODIAZEPINE DERIVATIVES AND THEIR USE AS CCK-MODULATORS GLAXO GROUP LTD (GB) 1998-07-08 EP disclosed
US-5569654-A ADMINISTERING AS ANTAGONISTS OF GASTRIN AND CHOLECYSTOKININ GLAXO GROUP LIMITED (GB) 1996-10-29 US disclosed