SCHEMBL8553824

SCHEMBL8553824

CN(C(=O)CN1C(=O)C(N)N=C(CN2CCOCC2)c2ccccc21)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.41
DRD4 P21917 1/20 0.40
ALDH1A1 P00352 4/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
ALDH3A1 P30838 1/20 0.37
OXTR P30559 1/20 0.37
LMNA P02545 2/20 0.36
HTT P42858 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
TP53 P04637 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
NPC1 O15118 1/20 0.35
CBLB Q13191 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8555248 0.87 OXTR (0.41) POLBDRD4OXTRCBLB
SCHEMBL8555947 0.84 HRH3 (0.38) POLBALDH1A1CA1CA2ALDH3A1
SCHEMBL8552793 0.83 CCKBR (0.48)
SCHEMBL9007270 0.83 CCKBR (0.39) POLBDRD4ALDH1A1LMNA
SCHEMBL8554964 0.81 ALDH1A1 (0.48) POLBALDH1A1CA1CA2ALDH3A1
SCHEMBL8552604 0.80 CCKBR (0.48)
SCHEMBL8552734 0.80 POLB (0.44) POLBALDH1A1LMNATP53
SCHEMBL9573635 0.78 GABRP (0.56) POLBOXTRTP53
SCHEMBL1388598 0.78 CCKBR (0.59)
SCHEMBL1388679 0.77 CCKBR (0.53)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0672037-B1 1,4-BENZODIAZEPINE DERIVATIVES AND THEIR USE AS CCK-MODULATORS GLAXO GROUP LTD (GB) 1998-07-08 EP disclosed
US-5569654-A ADMINISTERING AS ANTAGONISTS OF GASTRIN AND CHOLECYSTOKININ GLAXO GROUP LIMITED (GB) 1996-10-29 US disclosed