SCHEMBL8555052

SCHEMBL8555052

Cc1cccc(C)c1NC(=O)CN1CCN(C(C)c2nc(-c3ccccc3)c(-c3ccccc3)o2)CC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.45
CYP2D6 P10635 2/20 0.45
ADRB1 P08588 2/20 0.45
ADRA2A P08913 2/20 0.45
ADRA2B P18089 2/20 0.45
ADRA2C P18825 2/20 0.45
ADRA1A P35348 2/20 0.45
DRD3 P35462 2/20 0.45
HTR2B P41595 2/20 0.45
KCNH2 Q12809 2/20 0.45
TSHR P16473 1/20 0.45
NFKB1 P19838 1/20 0.45
ADRB2 P07550 1/20 0.45
SCN5A Q14524 1/20 0.45
LMNA P02545 3/20 0.44
BLM P54132 1/20 0.44
PMP22 Q01453 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
MEN1 O00255 4/20 0.44
KMT2A Q03164 4/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8555057 0.83 NR4A2 (0.51) CYP3A4CYP2D6ADRB1ADRA2AADRA2B
SCHEMBL8552887 0.83 NR4A2 (0.47) CYP3A4CYP2D6ADRB1ADRA2AADRA2B
SCHEMBL8558360 0.81 RXRA (0.50) CYP3A4CYP2D6ADRB1ADRA2AADRA2B
SCHEMBL8557576 0.75 MEN1 (0.52) CYP3A4CYP2D6ADRB1ADRA2AADRA2B
SCHEMBL8553475 0.74 GAA (0.45) CYP3A4CYP2D6ADRB1ADRA2AADRA2B
SCHEMBL2327539 0.73 ALDH1A1 (0.64) CYP3A4CYP2D6ADRB1ADRA2AADRA2B
SCHEMBL8557330 0.73 CETP (0.43) CYP3A4CYP2D6ADRB1ADRA2AADRA2B
Hydrochloric Acid SCHEMBL8554703 0.73 GAA (0.43) CYP3A4CYP2D6ADRB1ADRA2AADRA2B
SCHEMBL8556400 0.72 NR4A2 (0.41) CYP3A4ADRA1ADRD3TSHRLMNA
SCHEMBL8552938 0.72 RXRA (0.46) KCNH2KMT2AALDH1A1KDRRXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0582164-B1 Adenosine re-uptake inhibiting derivatives of diphenyl oxazoles, thiazoles and imidazoles BRISTOL MYERS SQUIBB CO (US) 1998-12-23 EP claimed
US-5382584-A Antiischemic agents BRISTOL-MYERS SQUIBB COMPANY (US) 1995-01-17 US claimed
EP-0582164-A1 Adenosine re-uptake inhibiting derivatives of diphenyl oxazoles, thiazoles and imidazoles Bristol-Myers Squibb Company (US) 1994-02-09 EP claimed