SCHEMBL8555844

SCHEMBL8555844

NC(N)=NS(=O)(=O)c1cnc(Cl)cc1Cl

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
F2 P00734 16/20 0.51
PRSS1 P07477 16/20 0.51
PRSS2 P07478 16/20 0.51
PRSS3 P35030 16/20 0.51
LMNA P02545 1/20 0.36
AGO2 Q9UKV8 1/20 0.36
ADRA2A P08913 1/20 0.35
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35
PLAU P00749 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8560220 0.73 F2 (0.47) F2PRSS1PRSS2PRSS3LMNA
SCHEMBL31584278 0.72 TRPV4 (0.40)
SCHEMBL23140985 0.72 TRPV4 (0.40)
SCHEMBL8555843 0.71 CA1 (0.32) F2PRSS1PRSS2PRSS3PLAU
SCHEMBL8558200 0.69 F2 (0.49) F2PRSS1PRSS2PRSS3LMNA
SCHEMBL10515229 0.68 F2 (0.59) F2PRSS1PRSS2PRSS3LMNA
SCHEMBL29799541 0.63 NNMT (0.61) LMNA
SCHEMBL384113 0.63 NNMT (0.61) LMNA
SCHEMBL8559284 0.62 CA1 (0.52) LMNA
SCHEMBL23833649 0.61 PDIA6 (0.41) LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0618209-B1 Pyridothiadiazines, processes for their preparation and pharmaceutical compositions containing them ADIR (FR) 1998-12-23 EP disclosed
US-5459138-A Dysfunctions of glutamatergic neurotransmission associated with learning and memory ADIR ET COMPAGNIE (FR) 1995-10-17 US disclosed
EP-0618209-A1 Pyridothiadiazines, processes for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1994-10-05 EP disclosed