SCHEMBL8555856

SCHEMBL8555856

CC(=O)c1cc(Br)ccc1OC(CC(C)O)c1cccnc1

nearest known ligand 0.53

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 9/20 0.53
HSD17B10 Q99714 1/20 0.43
PTGDR2 Q9Y5Y4 1/20 0.42
KMT2A Q03164 1/20 0.42
KCNA5 P22460 2/20 0.39
ADRB3 P13945 2/20 0.38
ADRB1 P08588 1/20 0.38
SORT1 Q99523 1/20 0.38
PDE4D Q08499 1/20 0.38
MKNK1 Q9BUB5 1/20 0.36
MKNK2 Q9HBH9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8071527 0.80 CYP3A4 (0.49) LRRK2KCNA5
SCHEMBL8186428 0.80 CYP3A4 (0.49) LRRK2KCNA5
SCHEMBL8553152 0.80 KCNA5 (0.47) LRRK2HSD17B10KMT2AKCNA5ADRB3
SCHEMBL7772046 0.78 SLC6A4 (0.42) LRRK2KMT2AKCNA5
SCHEMBL7773934 0.78 SLC6A4 (0.42) LRRK2KMT2AKCNA5
SCHEMBL8557113 0.74 CYP51A1 (0.47) KMT2AADRB3ADRB1PDE4DMKNK1
SCHEMBL8555243 0.71 AKR1C3 (0.41) KCNA5ADRB3ADRB1MKNK1MKNK2
SCHEMBL8555638 0.71 SUCNR1 (0.43) KMT2AKCNA5ADRB3ADRB1
SCHEMBL8554047 0.71 SLC6A2 (0.51) KCNA5
SCHEMBL8550969 0.70 EPHX1 (0.46) KCNA5ADRB3ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0865431-A2 COMPOUNDS Astra Pharmaceuticals Limited (GB) 1998-09-23 EP disclosed
WO-1997020815-A1 COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1997-06-12 WO disclosed