SCHEMBL8555900

SCHEMBL8555900

O=C(O)CN1C(=O)C(=O)[N]c2ccccc21

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.50
CA9 Q16790 2/20 0.50
APEX1 P27695 3/20 0.43
PTGES O14684 1/20 0.43
MEN1 O00255 4/20 0.41
KMT2A Q03164 4/20 0.41
AKR1B1 P15121 2/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP1A2 P05177 1/20 0.41
MAPT P10636 1/20 0.41
HPGD P15428 1/20 0.41
ALOX15 P16050 1/20 0.41
HSD17B10 Q99714 1/20 0.41
ATM Q13315 1/20 0.39
CA2 P00918 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6013595 0.78 ALDH1A1 (0.46) CA12CA9MEN1KMT2AKDM4E
SCHEMBL9618341 0.72 CA12 (0.65) CA12CA9APEX1PTGESMEN1
SCHEMBL9034857 0.72 AADAT (0.36) KDM4EALDH1A1
SCHEMBL30519490 0.71 CES1 (0.65) CA12CA9MEN1KMT2AALDH1A1
SCHEMBL3012558 0.71 CES1 (0.65) CA12CA9MEN1KMT2AALDH1A1
SCHEMBL2338193 0.69 ALDH1A1 (0.50) MEN1KMT2AALDH1A1MAPTHPGD
SCHEMBL29744481 0.67 CA12 (1.00) CA12CA9MEN1KMT2AAKR1B1
SCHEMBL522649 0.67 CA12 (1.00) CA12CA9MEN1KMT2AAKR1B1
SCHEMBL3373741 0.67 CA12 (0.53) CA12CA9APEX1MEN1KMT2A
SCHEMBL2228228 0.67 OPRL1 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0647137-A4 GLYCINE RECEPTOR ANTAGONISTS AND THE USE THEREOF. UNIV CALIFORNIA WEBER ECKARD (US) 1998-09-16 EP disclosed
EP-0647137-A1 GLYCINE RECEPTOR ANTAGONISTS AND THE USE THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1995-04-12 EP disclosed