SCHEMBL8556969

SCHEMBL8556969

O=C(CN1CCN(Cc2nc(-c3ccccc3)c(-c3ccccc3)o2)CC1)Nc1ccc(F)cc1

nearest known ligand 0.64

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
REV1 Q9UBZ9 1/20 0.53
ACHE P22303 1/20 0.52
BACE1 P56817 1/20 0.52
ALDH1A1 P00352 6/20 0.51
KDM4E B2RXH2 2/20 0.51
ATM Q13315 2/20 0.51
THRB P10828 1/20 0.51
OGA O60502 1/20 0.51
CHRNB2 P17787 2/20 0.49
CHRNB4 P30926 2/20 0.49
CHRNA3 P32297 2/20 0.49
CHRNA4 P43681 2/20 0.49
KMT2A Q03164 3/20 0.48
MAPT P10636 1/20 0.48
KDR P35968 1/20 0.48
TSHR P16473 1/20 0.47
MEN1 O00255 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8553993 0.93 KDR (0.54) ALDH1A1KDM4EATMTHRBOGA
SCHEMBL8554363 0.91 KDR (0.57) KDM4EATMOGAKMT2AKDR
SCHEMBL8555039 0.90 ATM (0.62) ACHEBACE1ALDH1A1KDM4EATM
SCHEMBL8557154 0.87 KDR (0.60) ALDH1A1KDM4EOGAKMT2AMAPT
SCHEMBL8557576 0.83 MEN1 (0.52) REV1ALDH1A1OGAKMT2ATSHR
SCHEMBL8552887 0.82 NR4A2 (0.47) ALDH1A1KDM4EKMT2AKDRTSHR
SCHEMBL8554568 0.82 KDR (0.58) ALDH1A1KDM4EATMKMT2AMAPT
SCHEMBL18409631 0.81 KCNH2 (0.49) ACHEALDH1A1KDM4EATMKMT2A
SCHEMBL8557836 0.79 SLC29A1 (0.43) ALDH1A1OGAKMT2AMAPTKDR
SCHEMBL8553599 0.79 KDR (0.48) ACHEALDH1A1KDM4EKMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0582164-B1 Adenosine re-uptake inhibiting derivatives of diphenyl oxazoles, thiazoles and imidazoles BRISTOL MYERS SQUIBB CO (US) 1998-12-23 EP claimed
US-5382584-A Antiischemic agents BRISTOL-MYERS SQUIBB COMPANY (US) 1995-01-17 US claimed
EP-0582164-A1 Adenosine re-uptake inhibiting derivatives of diphenyl oxazoles, thiazoles and imidazoles Bristol-Myers Squibb Company (US) 1994-02-09 EP claimed