SCHEMBL8555039

SCHEMBL8555039

O=C(CN1CCN(Cc2nc(-c3ccccc3)c(-c3ccccc3)o2)CC1)Nc1ccc(Cl)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.62
KDR P35968 4/20 0.58
RXRA P19793 2/20 0.52
RXRB P28702 2/20 0.52
RXRG P48443 2/20 0.52
ACHE P22303 1/20 0.52
BACE1 P56817 1/20 0.52
OGA O60502 1/20 0.51
MEN1 O00255 3/20 0.50
KMT2A Q03164 3/20 0.50
KCNA5 P22460 1/20 0.48
ALDH1A1 P00352 2/20 0.47
MAPT P10636 2/20 0.47
CACNA1G O43497 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA7 P43166 1/20 0.47
LMNA P02545 1/20 0.46
HTT P42858 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8553993 0.93 KDR (0.54) ATMKDRRXRARXRBRXRG
SCHEMBL8554363 0.91 KDR (0.57) ATMKDRRXRARXRBOGA
SCHEMBL8556969 0.90 REV1 (0.53) ATMKDRACHEBACE1OGA
SCHEMBL8557154 0.87 KDR (0.60) KDROGAMEN1KMT2AKCNA5
SCHEMBL8554568 0.86 KDR (0.58) ATMKDRRXRARXRBRXRG
SCHEMBL8553599 0.83 KDR (0.48) KDRRXRARXRBRXRGACHE
SCHEMBL8552887 0.82 NR4A2 (0.47) KDRRXRARXRBRXRGMEN1
SCHEMBL8554274 0.80 KDR (0.45) KDRACHEBACE1ALDH1A1MAPT
SCHEMBL18409351 0.79 ALDH1A1 (0.54) KDRRXRARXRBRXRGALDH1A1
SCHEMBL18409735 0.77 KCNH2 (0.58) RXRARXRBRXRGALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0582164-B1 Adenosine re-uptake inhibiting derivatives of diphenyl oxazoles, thiazoles and imidazoles BRISTOL MYERS SQUIBB CO (US) 1998-12-23 EP claimed
US-5382584-A Antiischemic agents BRISTOL-MYERS SQUIBB COMPANY (US) 1995-01-17 US claimed
EP-0582164-A1 Adenosine re-uptake inhibiting derivatives of diphenyl oxazoles, thiazoles and imidazoles Bristol-Myers Squibb Company (US) 1994-02-09 EP claimed