SCHEMBL8557086

SCHEMBL8557086

O=C1COc2cc([N+](=O)[O-])ccc2N1Cc1ccccc1Cl

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.67
CYP1A2 P05177 2/20 0.46
CYP2C19 P33261 2/20 0.46
CYP2C9 P11712 1/20 0.46
SLC5A1 P13866 1/20 0.45
SLC5A2 P31639 1/20 0.45
CYP2D6 P10635 1/20 0.44
MEN1 O00255 4/20 0.43
KMT2A Q03164 4/20 0.43
GAA P10253 2/20 0.43
HTT P42858 2/20 0.42
CASP1 P29466 1/20 0.41
CASP3 P42574 1/20 0.41
CASP4 P49662 1/20 0.41
CASP7 P55210 1/20 0.41
CASP9 P55211 1/20 0.41
CASP6 P55212 1/20 0.41
CASP8 Q14790 1/20 0.41
MAPT P10636 4/20 0.41
TP53 P04637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8553215 0.91 TSHR (0.67) TSHRCYP1A2CYP2C19CYP2C9SLC5A1
SCHEMBL27376595 0.86 CASP1 (0.56) TSHRCYP2C19CYP2C9SLC5A1SLC5A2
SCHEMBL8624433 0.83 SLC5A1 (0.51) TSHRSLC5A1SLC5A2CASP1CASP3
SCHEMBL29256246 0.83 TSHR (0.45) TSHRSLC5A1SLC5A2MEN1KMT2A
SCHEMBL27377925 0.81 SLC5A1 (0.48) TSHRCYP1A2CYP2C19CYP2C9SLC5A1
SCHEMBL27376612 0.80 CYP1A2 (0.56) TSHRCYP1A2CYP2C19CYP2C9CYP2D6
SCHEMBL30806430 0.80 CYP1A2 (0.56) TSHRCYP1A2CYP2C19CYP2C9CYP2D6
SCHEMBL9687134 0.79 BRD4 (0.50) TSHRSLC5A1SLC5A2MEN1KMT2A
SCHEMBL282621 0.79 TERT (0.44) SLC5A1SLC5A2MEN1KMT2AGAA
SCHEMBL8130592 0.78 TERT (0.48) TSHRCYP1A2SLC5A1SLC5A2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0869949-A1 BENZOXAZINE ANTIMICROBIAL AGENTS ORTHO PHARMACEUTICAL CORPORATION (US) 1998-10-14 EP disclosed
WO-1997017333-A1 BENZOXAZINE ANTIMICROBIAL AGENTS ORTHO PHARMACEUTICAL CORPORATION (US) 1997-05-15 WO disclosed