SCHEMBL8558762

SCHEMBL8558762

CCN(c1ccccc1)S(=O)(=O)c1ccc2c(c1)CCC(C)(C)O2

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DAGLA Q9Y4D2 9/20 0.56
CYP3A4 P08684 2/20 0.56
CYP2D6 P10635 2/20 0.56
CYP2C9 P11712 2/20 0.56
CYP2C19 P33261 2/20 0.56
KCNH2 Q12809 2/20 0.56
ABHD6 Q9BV23 2/20 0.54
HIF1A Q16665 1/20 0.52
EPAS1 Q99814 1/20 0.52
ESR1 P03372 2/20 0.49
TSHR P16473 1/20 0.48
MAPK1 P28482 1/20 0.48
KMT2A Q03164 1/20 0.48
HSD17B10 Q99714 1/20 0.48
PKM P14618 2/20 0.47
PKLR P30613 1/20 0.47
ALPL P05186 1/20 0.47
ALPI P09923 1/20 0.47
MAPT P10636 1/20 0.47
ALPG P10696 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8557971 0.85 ATM (0.56) DAGLACYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL8487793 0.82 DAGLA (0.59) DAGLACYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL7821527 0.77 ESR1 (0.46) HIF1AEPAS1ESR1TSHRMAPK1
SCHEMBL12355590 0.75 DAGLA (0.87) DAGLACYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL8557486 0.75 DAGLA (0.49) DAGLACYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL3380011 0.75 DAGLA (0.55) DAGLACYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL2242243 0.74 DAGLA (0.53) DAGLACYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL8553826 0.74 DAGLA (0.51) DAGLACYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL8557904 0.74 PKM (0.73) DAGLACYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL7812015 0.74 HIF1A (0.69) HIF1AEPAS1ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1185153-A Benzopyrans and pharmaceutical composition contg. same CIBA GEIGY AG (CH) 1998-06-17 CN disclosed
EP-0828733-A1 BENZOPYRANS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Novartis AG (CH) 1998-03-18 EP disclosed
WO-1996037490-A1 BENZOPYRANS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM NOVARTIS AG (CH) 1996-11-28 WO disclosed