SCHEMBL8554274

SCHEMBL8554274

O=C(CN1CCN(Cc2nc(-c3ccccc3)c(-c3ccccc3)o2)CC1)Nc1c(Cl)cc([N+](=O)[O-])cc1Cl

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 2/20 0.45
ACHE P22303 1/20 0.45
BACE1 P56817 1/20 0.45
DYRK1A Q13627 1/20 0.45
ALDH1A1 P00352 8/20 0.42
MAPT P10636 3/20 0.42
GAA P10253 2/20 0.42
LMNA P02545 2/20 0.42
HTT P42858 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
DRD4 P21917 1/20 0.41
NR4A2 P43354 2/20 0.40
NR4A1 P22736 1/20 0.40
NR4A3 Q92570 1/20 0.40
KDM4E B2RXH2 1/20 0.40
GFER P55789 1/20 0.40
MCL1 Q07820 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8553599 0.88 KDR (0.48) KDRACHEALDH1A1MAPTGAA
SCHEMBL8554568 0.87 KDR (0.58) KDRALDH1A1MAPTGAALMNA
SCHEMBL8414147 0.87 SLC29A1 (0.43) KDRACHEBACE1DYRK1ALMNA
Hydrochloric Acid SCHEMBL8595835 0.86 SLC29A1 (0.43) KDRACHEBACE1DYRK1AALDH1A1
SCHEMBL8553993 0.80 KDR (0.54) KDRALDH1A1LMNASMN1; SMN2NPC1
SCHEMBL8555039 0.80 ATM (0.62) KDRACHEBACE1ALDH1A1MAPT
SCHEMBL8552887 0.80 NR4A2 (0.47) KDRALDH1A1LMNANR4A2NR4A1
SCHEMBL8557836 0.79 SLC29A1 (0.43) KDRALDH1A1MAPTGAALMNA
SCHEMBL8554363 0.77 KDR (0.57) KDRLMNAHTTNR4A2KDM4E
SCHEMBL8556969 0.76 REV1 (0.53) KDRACHEBACE1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0582164-B1 Adenosine re-uptake inhibiting derivatives of diphenyl oxazoles, thiazoles and imidazoles BRISTOL MYERS SQUIBB CO (US) 1998-12-23 EP claimed
EP-0582164-A1 Adenosine re-uptake inhibiting derivatives of diphenyl oxazoles, thiazoles and imidazoles Bristol-Myers Squibb Company (US) 1994-02-09 EP claimed