SCHEMBL855805

SCHEMBL855805

CN(C(=O)O)c1nc2cnc(Br)cc2[nH]1

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 4/20 0.33
HTT P42858 1/20 0.31
HSP90AA1 P07900 1/20 0.31
ESR2 Q92731 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
PIN1 Q13526 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5897147 0.76 HSD17B10 (0.48) TDP1
SCHEMBL251109 0.74 LMNA (0.53) HTTTDP1
SCHEMBL544668 0.74 SMAD3 (0.41) HTT
SCHEMBL11436852 0.74 PIN1 (0.59) HTTHSP90AA1ESR2TDP1PIN1
SCHEMBL3715874 0.71 NPC1 (0.42)
SCHEMBL11096785 0.69 TDP1 (0.35) MCHR1HTTHSP90AA1ESR2TDP1
SCHEMBL830501 0.69 KDM4E (0.34) HTTTDP1
SCHEMBL3388847 0.69 ALDH1A1 (0.65) HTT
SCHEMBL4279399 0.69 HPGD (0.51) HTT
SCHEMBL11118273 0.68 LMNA (0.57) MCHR1HSP90AA1ESR2TDP1PIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2432779-A1 BENZOXAZEPINES BASED P13K/MT0R INHIBITORS AGAINST PROLIFERATIVE DISEASES Exelixis, Inc. (US) 2012-03-28 EP disclosed