SCHEMBL8558088

SCHEMBL8558088

CCC(OC1CCCOC1)C1CC(c2ccc(Cl)c(Cl)c2)CN(Cc2ccccc2)C1=O

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 3/20 0.39
OPRM1 P35372 3/20 0.36
OPRK1 P41145 3/20 0.36
PDE4B Q07343 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35
SLC6A3 Q01959 3/20 0.34
TACR1 P25103 1/20 0.33
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
KCNH2 Q12809 1/20 0.32
SIGMAR1 Q99720 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8300797 0.90 PDE4A (0.40) PDE4AOPRM1OPRK1PDE4BPDE4C
SCHEMBL8291779 0.71 SLC6A4 (0.43) SLC6A3SLC6A2SLC6A4KCNH2
SCHEMBL8292203 0.71 UTS2R (0.41) OPRM1OPRK1SLC6A3TACR1SLC6A4
SCHEMBL8298259 0.71 SLC6A2 (0.36) OPRM1OPRK1SLC6A3SLC6A2SLC6A4
SCHEMBL7846543 0.69 TACR1 (0.47) TACR1
SCHEMBL8564881 0.69 PDE4A (0.38) PDE4APDE4BPDE4CPDE4D
SCHEMBL8291783 0.69 SLC6A2 (0.41) SLC6A3SLC6A2SLC6A4KCNH2
SCHEMBL8311113 0.69 SLC6A2 (0.44) PDE4BSLC6A3SLC6A2SLC6A4KCNH2
SCHEMBL8300632 0.68 SLC6A2 (0.46) SLC6A3SLC6A2SLC6A4KCNH2
SCHEMBL8292045 0.68 SLC6A2 (0.38) SLC6A3SLC6A2SLC6A4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5807865-A 3,3-disubstituted piperidine derivatives and their use as therapeutic agents MERCK SHARP & DOHME LIMITED (GB) 1998-09-15 US disclosed