SCHEMBL8298259

SCHEMBL8298259

CCC(OC1CCCOC1)N1CC(c2ccc(Cl)c(Cl)c2)CCC1=O

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 6/20 0.36
SLC6A4 P31645 6/20 0.36
SLC6A3 Q01959 6/20 0.36
KCNH2 Q12809 4/20 0.36
SRD5A1 P18405 1/20 0.33
ENPP2 Q13822 3/20 0.33
P2RX7 Q99572 1/20 0.31
CYP2D6 P10635 4/20 0.31
KCNA5 P22460 1/20 0.30
SCN5A Q14524 1/20 0.30
CXCR2 P25025 1/20 0.30
OPRM1 P35372 1/20 0.30
OPRK1 P41145 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8292045 0.88 SLC6A2 (0.38) SLC6A2SLC6A4SLC6A3KCNH2SRD5A1
SCHEMBL8291779 0.82 SLC6A4 (0.43) SLC6A2SLC6A4SLC6A3KCNH2CYP2D6
SCHEMBL8291783 0.74 SLC6A2 (0.41) SLC6A2SLC6A4SLC6A3KCNH2CYP2D6
SCHEMBL8311113 0.73 SLC6A2 (0.44) SLC6A2SLC6A4SLC6A3KCNH2CYP2D6
SCHEMBL8300632 0.73 SLC6A2 (0.46) SLC6A2SLC6A4SLC6A3KCNH2CYP2D6
SCHEMBL8558088 0.71 PDE4A (0.39) SLC6A2SLC6A4SLC6A3KCNH2OPRM1
SCHEMBL8300797 0.69 PDE4A (0.40) SLC6A2SLC6A4SLC6A3KCNH2KCNA5
SCHEMBL7172151 0.65 IDH1 (0.35)
SCHEMBL8204373 0.64 SLC6A3 (0.39) SLC6A2SLC6A4SLC6A3
SCHEMBL7846543 0.64 TACR1 (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0512901-B1 Aminated polycyclic compounds and their enantiomers, process for their preparation and pharmaceutical compositions containing them SANOFI SA (FR) 1999-06-23 EP claimed
US-5807865-A 3,3-disubstituted piperidine derivatives and their use as therapeutic agents MERCK SHARP & DOHME LIMITED (GB) 1998-09-15 US disclosed