SCHEMBL8558206

SCHEMBL8558206

CC[C@H](C)[C@H](NC(=O)Cc1ccc(Cl)cc1C)C(=O)OC

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 4/20 0.52
NOS1 P29475 4/20 0.52
NOS2 P35228 4/20 0.52
ALDH1A1 P00352 6/20 0.51
HTT P42858 1/20 0.51
POLB P06746 2/20 0.46
MAPT P10636 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
TAS1R3 Q7RTX0 1/20 0.45
TAS1R1 Q7RTX1 1/20 0.45
CACNA1H O95180 2/20 0.43
MEN1 O00255 1/20 0.42
LMNA P02545 1/20 0.42
KMT2A Q03164 1/20 0.42
KDM4E B2RXH2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8652110 1.00 NOS3 (0.52) NOS3NOS1NOS2ALDH1A1HTT
SCHEMBL8557162 0.89 ALDH1A1 (0.57) ALDH1A1HTTNPSR1TAS1R3TAS1R1
SCHEMBL8657482 0.89 ALDH1A1 (0.57) ALDH1A1HTTNPSR1TAS1R3TAS1R1
SCHEMBL8558470 0.88 FPR2 (0.44) ALDH1A1MEN1KMT2AKDM4E
SCHEMBL8558467 0.88 FPR2 (0.44) ALDH1A1MEN1KMT2AKDM4E
SCHEMBL6475338 0.87 NOS3 (0.51) NOS3NOS1NOS2ALDH1A1HTT
SCHEMBL4425149 0.87 NOS3 (0.51) NOS3NOS1NOS2ALDH1A1HTT
SCHEMBL7964516 0.87 ALDH1A1 (0.56) NOS3NOS1NOS2ALDH1A1HTT
SCHEMBL6996770 0.87 ALDH1A1 (0.56) NOS3NOS1NOS2ALDH1A1HTT
SCHEMBL8553227 0.84 ALDH1A1 (0.55) NOS3NOS1NOS2ALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1080719-C Substituted 1H-3-aryl-pyrrolidine-2,4-diones derivative BAYER GMBH (DE) 2002-03-13 CN disclosed
US-5847211-A Substituted 1H-3-Aryl-pyrrolidine-2,4-dione derivatives BAYER AKTIENGESELLSCHAFT (DE) 1998-12-08 US disclosed
EP-0668267-B1 Substituted 1H-3-aryl-pyrrolidine-2,4-dione derivatives BAYER AG (DE) 1998-04-08 EP disclosed
US-5622917-A PESTICIDES BAYER AKTIENGESELLSCHAFT (DE) 1997-04-22 US disclosed
CN-1110680-A Substituted 1H-3-aryl-pyrrolidine-2,4-diones derivative BYLL GMBH (DE) 1995-10-25 CN disclosed
EP-0668267-A1 Substituted 1H-3-aryl-pyrrolidine-2,4-dione derivatives BAYER AG (DE) 1995-08-23 EP disclosed