SCHEMBL8558377

SCHEMBL8558377

COc1ccc(NC(=O)c2ccc(C(=O)N3Cc4ccccc4Cc4ccccc43)cc2)cc1Cl

nearest known ligand 0.59

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 3/20 0.54
NPC1 O15118 4/20 0.52
RAB9A P51151 4/20 0.52
SMN1; SMN2 Q16637 4/20 0.52
MAPT P10636 2/20 0.52
KDM4E B2RXH2 1/20 0.52
TP53 P04637 1/20 0.52
HSD17B10 Q99714 1/20 0.52
AVPR2 P30518 1/20 0.51
AVPR1A P37288 1/20 0.51
ACHE P22303 3/20 0.50
HSD17B3 P37058 1/20 0.50
ATM Q13315 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8561097 0.85 AVPR2 (0.52) NAMPTNPC1RAB9ASMN1; SMN2MAPT
SCHEMBL8557743 0.83 AVPR2 (0.64) AVPR2AVPR1AACHE
SCHEMBL8557503 0.82 ACHE (0.58) NPC1RAB9ASMN1; SMN2AVPR2AVPR1A
SCHEMBL8563019 0.82 AVPR2 (0.59) NAMPTAVPR2AVPR1AACHE
SCHEMBL8558857 0.82 HPGD (0.57) NAMPTNPC1RAB9ASMN1; SMN2
SCHEMBL8560873 0.81 ACHE (0.60) NAMPTRAB9AAVPR2AVPR1AACHE
SCHEMBL8563565 0.81 NAMPT (0.50) NAMPTNPC1RAB9ASMN1; SMN2MAPT
SCHEMBL8559349 0.81 AVPR2 (0.60) AVPR2AVPR1AACHE
SCHEMBL8556252 0.80 NAMPT (0.63) NAMPTNPC1RAB9ASMN1; SMN2MAPT
SCHEMBL8558993 0.79 AVPR2 (0.65) AVPR2AVPR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640592-B1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID CO (US) 1998-12-30 EP disclosed