SCHEMBL8558917

SCHEMBL8558917

CCOC(C=O)c1ccc2c(c1)CC(n1ccnc1C(=O)O)C2=O

nearest known ligand 0.30

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.30
PTGS2 P35354 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8558748 0.77 METAP1 (0.39) ACHE
SCHEMBL7834401 0.77 TBXAS1 (0.36)
SCHEMBL8557548 0.75 METAP1 (0.38)
SCHEMBL8555982 0.75 METAP1 (0.38)
SCHEMBL8880656 0.73 METAP1 (0.38)
SCHEMBL8558771 0.72 KDM4E (0.40) ACHE
SCHEMBL8880563 0.71 GABRG2 (0.38)
SCHEMBL8881385 0.71 GABRG2 (0.41)
SCHEMBL8881176 0.71 CYP19A1 (0.43)
SCHEMBL8090657 0.70 GABRA1 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0820455-A1 5H, 10H-IMIDAZO [1,2-a]INDENO [1,2-e]PYRAZIN-4-ONE DERIVATIVES, PREPARATION THEREOF, AND DRUGS CONTAINING SAID DERIVATIVES Aventis Pharma S.A. (FR) 1998-01-28 EP disclosed
WO-1996031511-A1 5H,10H-IMIDAZO[1,2-a]INDENO[1,2-e]PYRAZIN-4-ONE DERIVATIVES, PREPARATION THEREOF, AND DRUGS CONTAINING SAID DERIVATIVES RHONE-POULENC RORER S.A. (FR) 1996-10-10 WO disclosed