SCHEMBL8559023

SCHEMBL8559023

Oc1ccc2c(CCCCN3CCC(c4c[nH]c5ccc(O)cc45)CC3)c[nH]c2c1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.60
CYP3A4 P08684 2/20 0.60
CYP2C9 P11712 2/20 0.60
CYP2D6 P10635 1/20 0.60
THPO P40225 1/20 0.60
MAPT P10636 2/20 0.52
BLM P54132 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
HTR1A P08908 2/20 0.52
DRD2 P14416 2/20 0.52
DRD3 P35462 2/20 0.52
TSHR P16473 1/20 0.52
DRD4 P21917 1/20 0.52
CYP2C19 P33261 1/20 0.52
TDP1 Q9NUW8 1/20 0.52
CCR2 P41597 2/20 0.51
HTR1B P28222 1/20 0.51
HTR2A P28223 1/20 0.51
HTR2C P28335 1/20 0.51
HTR1E P28566 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8559641 0.95 CYP1A2 (0.63) CYP1A2CYP3A4CYP2C9CYP2D6THPO
SCHEMBL8556970 0.93 ADRA1D (0.60) CYP1A2CYP3A4CYP2C9CYP2D6THPO
SCHEMBL8554847 0.91 CYP1A2 (0.65) CYP1A2CYP3A4CYP2C9CYP2D6THPO
SCHEMBL8556284 0.91 HTR1A (0.57) CYP1A2CYP3A4CYP2C9CYP2D6THPO
SCHEMBL8559411 0.90 HTR1A (0.61) CYP1A2CYP3A4CYP2C9CYP2D6THPO
SCHEMBL8558927 0.89 ADRA1D (0.63) CYP1A2CYP3A4CYP2C9MAPTHTR1A
SCHEMBL8553229 0.86 HTR1A (0.64) HTR1ADRD2HTR2AHTR7HTR6
SCHEMBL11357559 0.84 DRD2 (0.54) CYP1A2CYP3A4CYP2C9CYP2D6MAPT
SCHEMBL7533678 0.84 CYP1A2 (0.61) CYP1A2CYP3A4CYP2C9CYP2D6THPO
SCHEMBL8558241 0.83 HTR1A (0.69) CYP1A2CYP3A4CYP2C9CYP2D6THPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0683166-B1 3-Indolylpiperidines MERCK PATENT GMBH (DE) 1998-10-28 EP disclosed