SCHEMBL8559319

SCHEMBL8559319

CN1CCc2cc(N3C(=O)NCC3c3ccccc3CCC(=O)O)ccc2C1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TMEM97 Q5BJF2 3/20 0.36
SIGMAR1 Q99720 3/20 0.36
PARP1 P09874 6/20 0.35
S1PR5 Q9H228 1/20 0.34
MAOA P21397 2/20 0.34
MAOB P27338 2/20 0.34
DRD1 P21728 2/20 0.34
DRD5 P21918 2/20 0.34
CRBN Q96SW2 1/20 0.34
PRMT5 O14744 1/20 0.34
WDR77 Q9BQA1 1/20 0.34
PTK2 Q05397 1/20 0.34
DRD2 P14416 1/20 0.33
DRD4 P21917 1/20 0.33
DRD3 P35462 1/20 0.33
KEAP1 Q14145 1/20 0.33
NFE2L2 Q16236 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8559857 0.97 PARP1 (0.36) TMEM97SIGMAR1PARP1DRD1DRD5
SCHEMBL8562403 0.87 HTR6 (0.40) PARP1DRD1DRD2
SCHEMBL8559323 0.83 PARP1 (0.37) TMEM97SIGMAR1PARP1
SCHEMBL8557053 0.83 HTR6 (0.41) PARP1PTK2
SCHEMBL8560491 0.82 HTR6 (0.43) PARP1
SCHEMBL8564812 0.80 ESR1 (0.31)
SCHEMBL8559860 0.80 PARP1 (0.39) SIGMAR1PARP1
Hydrochloric Acid SCHEMBL8563477 0.79 PARP1 (0.38) SIGMAR1PARP1
SCHEMBL8573544 0.74 P2RX3 (0.35)
Hydrochloric Acid SCHEMBL8560445 0.73 QPCT (0.39) TMEM97SIGMAR1PARP1DRD1KEAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5827849-A HAVING INHIBITORY EFFECT ON INFLAMMATION AND BONE DEGRADATION, ANTITHROMBOTIC, ANTIAGGREGATORY AND TUMOR- OR METASTASIS-INHIBITING EFFECT KARL THOMAE GMBH (DE) 1998-10-27 US disclosed