SCHEMBL8559738

SCHEMBL8559738

CCc1c(N2CCN(CC)CC2)c(F)cc2c(=O)c(OC(=O)O)c[nH]c12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 10/20 0.39
ALDH1A1 P00352 7/20 0.39
HSD17B10 Q99714 7/20 0.39
HPGD P15428 6/20 0.39
LMNA P02545 3/20 0.39
MAPT P10636 2/20 0.39
PMP22 Q01453 1/20 0.34
DRD3 P35462 1/20 0.33
BRD4 O60885 1/20 0.33
TSHR P16473 1/20 0.33
HTT P42858 1/20 0.33
CYP2J2 P51589 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
KMT2A Q03164 1/20 0.33
FGFR1 P11362 1/20 0.32
FGFR2 P21802 1/20 0.32
ADRA2B P18089 1/20 0.32
MAPK1 P28482 1/20 0.32
CYP2C9 P11712 1/20 0.32
ATP6V1B2 P21281 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4758703 0.92 KDM4E (0.38) KDM4EALDH1A1HSD17B10HPGDLMNA
SCHEMBL5507782 0.86 KDM4E (0.41) KDM4EALDH1A1HSD17B10HPGDLMNA
SCHEMBL9626409 0.79 KDM4E (0.40) KDM4EALDH1A1HSD17B10HPGDLMNA
SCHEMBL6673792 0.78 CYP1A2 (0.34) KDM4EALDH1A1HPGDLMNAKMT2A
SCHEMBL10696786 0.76 HTR6 (0.34) KDM4EALDH1A1HPGD
SCHEMBL5043939 0.76 KDM4E (0.50) KDM4EALDH1A1HSD17B10HPGDLMNA
SCHEMBL10610892 0.75 KDM4E (0.42) KDM4EALDH1A1HSD17B10HPGDLMNA
SCHEMBL5736019 0.74 KDM4E (0.41) KDM4EALDH1A1HSD17B10HPGDLMNA
SCHEMBL10707395 0.74 KDM4E (0.47) KDM4EALDH1A1HSD17B10HPGDLMNA
SCHEMBL10709201 0.72 KDM4E (0.46) KDM4EALDH1A1HSD17B10HPGDLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0828715-A1 N-OXIDES AS ANTIBACTERIAL AGENTS BAYER AG (DE) 1998-03-18 EP disclosed
WO-1996038417-A1 N-OXIDES AS ANTIBACTERIAL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 1996-12-05 WO disclosed