SCHEMBL8559784

SCHEMBL8559784

CC(C)c1ccc(C(=O)O)cc1C(=O)C(F)(F)F

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PLA2G2D Q9UNK4 1/20 0.54
ACE2 Q9BYF1 4/20 0.53
CES1 P23141 1/20 0.43
MLYCD O95822 4/20 0.42
BCL2 P10415 2/20 0.42
MCL1 Q07820 2/20 0.42
HDAC1 Q13547 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
GRM1 Q13255 2/20 0.41
MEN1 O00255 1/20 0.41
CYP1A2 P05177 1/20 0.41
KMT2A Q03164 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
KDM4E B2RXH2 1/20 0.40
RXRA P19793 2/20 0.40
RXRB P28702 1/20 0.40
RXRG P48443 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8558231 0.83 NOTUM (0.46) MLYCDKDM4E
SCHEMBL1355684 0.83 ACE2 (0.67) ACE2BCL2MCL1GRM1MEN1
SCHEMBL7009458 0.80 ACE2 (0.58) ACE2BCL2MCL1GRM1MEN1
SCHEMBL5874054 0.77 ACE2 (0.51) ACE2GRM1MEN1CYP1A2KMT2A
SCHEMBL8558758 0.76 PLA2G2D (0.55) PLA2G2DCES1HDAC1HDAC6MEN1
SCHEMBL13768197 0.76 MLYCD (0.50) CES1MLYCD
SCHEMBL32665932 0.75 CES1 (0.47) PLA2G2DCES1MLYCDBCL2MCL1
SCHEMBL13129171 0.75 CES1 (0.47) PLA2G2DCES1MLYCDBCL2MCL1
SCHEMBL8506645 0.75 ACE2 (0.50) ACE2GRM1MEN1CYP1A2KMT2A
SCHEMBL2159198 0.75 ACE2 (0.54) ACE2GRM1KDM4ERXRARXRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5747541-A Substituted benzoylguanidines, a process for their preparation, their use as medicament of diagnostic agent, and medicament comprising them HOECHST AKTIENGESELLSCHAFT (DE) 1998-05-05 US disclosed
EP-0765868-A1 Substituted bezoyl guanidines, process for their preparation, their use as antiarrhythmics or diagnostic agent as well as pharmaceuticals containing them HOECHST AKTIENGESELLSCHAFT (DE) 1997-04-02 EP disclosed