SCHEMBL8560283

SCHEMBL8560283

C=CCOc1ccc(CCC)c2c1C(C)(C)C(=O)N2

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.37
ALDH1A1 P00352 3/20 0.37
MAPT P10636 1/20 0.37
HPGD P15428 1/20 0.37
PDK2 Q15119 1/20 0.37
PDE4B Q07343 2/20 0.34
PDE4A P27815 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34
CYP3A4 P08684 1/20 0.33
CYP2A6 P11509 1/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA9 Q16790 1/20 0.33
TSHR P16473 3/20 0.32
CTSL P07711 1/20 0.32
CTSS P25774 1/20 0.32
CTSK P43235 1/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8556692 0.93 KDM4E (0.36) KDM4EALDH1A1MAPTHPGDPDK2
SCHEMBL8557800 0.92 KDM4E (0.35) KDM4EALDH1A1MAPTHPGDPDK2
SCHEMBL8557627 0.91 PDK2 (0.46) KDM4EALDH1A1MAPTHPGDPDK2
SCHEMBL8557767 0.91 THRA (0.36) KDM4EALDH1A1MAPTHPGDPDK2
SCHEMBL8555134 0.82 ALDH1A1 (0.37) KDM4EALDH1A1MAPTHPGDPDK2
SCHEMBL8555625 0.73 CYP3A4 (0.43) KDM4EALDH1A1MAPTHPGDPDK2
SCHEMBL8557831 0.73 ALDH1A1 (0.36) KDM4EALDH1A1MAPTHPGDPDK2
SCHEMBL8556960 0.73 PDK2 (0.44) PDK2
SCHEMBL8555928 0.69 PDK2 (0.35) PDK2
SCHEMBL8554583 0.67 PDE4B (0.37) KDM4EALDH1A1HPGDPDE4BCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0653426-B1 Indole derivatives, salts thereof and heart affection therapeutic agent comprising the same KOWA CO (JP) 1998-07-22 EP disclosed
US-5510366-A INOTROPIC, ANTIARRHYMTHMIA AGENTS, VASODILATORS KOWA CO., LTD. (JP) 1996-04-23 US disclosed
EP-0653426-A1 Indole derivatives, salts thereof and heart affection therapeutic agent comprising the same KOWA COMPANY, LTD. (JP) 1995-05-17 EP disclosed