SCHEMBL8560730

SCHEMBL8560730

O=C(Cc1cccs1)Nc1ccc(C(=O)N2Cc3ccccc3Sc3ccccc32)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 8/20 0.53
MEN1 O00255 6/20 0.53
KMT2A Q03164 6/20 0.53
NPC1 O15118 4/20 0.53
RAB9A P51151 4/20 0.53
BLM P54132 2/20 0.53
SMN1; SMN2 Q16637 2/20 0.49
MAPT P10636 1/20 0.48
CTDSP1 Q9GZU7 2/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
ALDH1A1 P00352 1/20 0.46
PKM P14618 1/20 0.46
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA5A P35218 1/20 0.46
CA7 P43166 1/20 0.46
CA9 Q16790 1/20 0.46
CA13 Q8N1Q1 1/20 0.46
CA5B Q9Y2D0 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8555635 0.85 HSD11B1 (0.47) MEN1KMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL9234962 0.83 AVPR1A (0.49) MEN1KMT2AAVPR2AVPR1A
SCHEMBL8559361 0.83 ALDH1A1 (0.44) MEN1KMT2ASMN1; SMN2MAPTALDH1A1
SCHEMBL8557995 0.82 KCNJ5 (0.47) THRBAVPR2AVPR1ANAMPT
SCHEMBL8556932 0.82 AVPR2 (0.48) POLBMEN1KMT2AMAPTAVPR2
SCHEMBL8557423 0.80 ACHE (0.51) RAB9AAVPR2AVPR1A
SCHEMBL8562542 0.77 AVPR1A (0.57) MEN1KMT2APKMAVPR2AVPR1A
SCHEMBL8563237 0.77 AVPR1A (0.59) AVPR2AVPR1A
SCHEMBL8556946 0.76 AVPR2 (0.55) AVPR2AVPR1A
SCHEMBL8559312 0.76 AVPR1A (0.55) AVPR2AVPR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640592-B1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID CO (US) 1998-12-30 EP disclosed
EP-0640592-A1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID COMPANY (US) 1995-03-01 EP disclosed