SCHEMBL8560824

SCHEMBL8560824

Clc1cc2[nH][c]nc2c(Cl)c1Cc1ccccc1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYMP P19971 1/20 0.34
SIRT2 Q8IXJ6 1/20 0.34
SIRT1 Q96EB6 1/20 0.34
CCNB2 O95067 2/20 0.33
CDK1 P06493 2/20 0.33
CCNB1 P14635 2/20 0.33
GSK3A P49840 2/20 0.33
GSK3B P49841 2/20 0.33
CCNB3 Q8WWL7 2/20 0.33
ALDH1A1 P00352 2/20 0.33
MEN1 O00255 1/20 0.33
MAPT P10636 1/20 0.33
KMT2A Q03164 1/20 0.33
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33
NR1H2 P55055 1/20 0.31
NR1H3 Q13133 1/20 0.31
PTGES O14684 1/20 0.31
CYP2C9 P11712 1/20 0.31
CALM1 P0DP23 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8558658 0.79 CCNB2 (0.37) TYMPSIRT2SIRT1CCNB2CDK1
SCHEMBL28514503 0.75 HPGD (0.33) ALDH1A1MEN1KMT2A
SCHEMBL433019 0.68 CYP3A4 (0.42) ALDH1A1MEN1KMT2ACYP2C9CALM1
SCHEMBL8562960 0.68 TUBB4A (0.37) CCNB2CDK1CCNB1GSK3AGSK3B
SCHEMBL8563998 0.67 IKBKB (0.36) PTGES
SCHEMBL10832750 0.66 MEN1 (0.30) MEN1MAPTKMT2A
SCHEMBL7617376 0.65 HTT (0.30)
SCHEMBL5319581 0.65 HTT (0.45) ALDH1A1MEN1MAPTKMT2AOPRM1
SCHEMBL29067648 0.64 TYMP (0.38) TYMPSIRT2SIRT1ALDH1A1MEN1
SCHEMBL11523704 0.64 CALM1 (0.58) TYMPALDH1A1MEN1KMT2AOPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0821675-A1 NOVEL HYDROXAMIC ACID AND AMINO-CARBOXYLATE COMPOUNDS AS METALLOPROTEASE AND TNF INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1998-02-04 EP disclosed
WO-1996033176-A1 NOVEL HYDROXAMIC ACID AND AMINO-CARBOXYLATE COMPOUNDS AS METALLOPROTEASE AND TNF INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-10-24 WO disclosed