SCHEMBL8558658

SCHEMBL8558658

Clc1ccc2[nH][c]nc2c1Cc1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNB2 O95067 2/20 0.37
CDK1 P06493 2/20 0.37
CCNB1 P14635 2/20 0.37
GSK3A P49840 2/20 0.37
GSK3B P49841 2/20 0.37
CCNB3 Q8WWL7 2/20 0.37
TYMP P19971 1/20 0.36
SIRT2 Q8IXJ6 1/20 0.35
SIRT1 Q96EB6 1/20 0.35
ALDH1A1 P00352 3/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
MAPT P10636 1/20 0.35
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
NR1H2 P55055 2/20 0.33
NR1H3 Q13133 1/20 0.33
CALM1 P0DP23 1/20 0.32
OPRM1 P35372 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8560824 0.79 TYMP (0.34) CCNB2CDK1CCNB1GSK3AGSK3B
SCHEMBL8562960 0.78 TUBB4A (0.37) CCNB2CDK1CCNB1GSK3AGSK3B
SCHEMBL10832750 0.71 MEN1 (0.30) MEN1KMT2AMAPTTDP1GAA
SCHEMBL8564117 0.70 CCNB2 (0.41) CCNB2CDK1CCNB1GSK3AGSK3B
SCHEMBL5247984 0.66 CALM1 (0.52) TYMPALDH1A1MEN1KMT2ATSHR
SCHEMBL7464217 0.65 CALM1 (0.46) CCNB2CDK1CCNB1GSK3AGSK3B
SCHEMBL8563838 0.65 SIRT1 (0.30) SIRT1
SCHEMBL11711485 0.64 CALM1 (0.44) TYMPALDH1A1MEN1KMT2AMAPT
SCHEMBL9790331 0.63 MEN1 (0.50) TYMPALDH1A1MEN1KMT2ACALM1
SCHEMBL11523704 0.61 CALM1 (0.58) TYMPALDH1A1MEN1KMT2ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0821675-A1 NOVEL HYDROXAMIC ACID AND AMINO-CARBOXYLATE COMPOUNDS AS METALLOPROTEASE AND TNF INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1998-02-04 EP disclosed
WO-1996033176-A1 NOVEL HYDROXAMIC ACID AND AMINO-CARBOXYLATE COMPOUNDS AS METALLOPROTEASE AND TNF INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-10-24 WO disclosed