SCHEMBL8556503

SCHEMBL8556503

c1ccc(CN2CCN(Cc3ncsn3)CC2)cc1

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 7/20 0.58
ALDH1A1 P00352 2/20 0.51
MC4R P32245 1/20 0.50
DRD4 P21917 2/20 0.49
POLB P06746 2/20 0.49
LMNA P02545 1/20 0.49
DRD2 P14416 1/20 0.47
DRD3 P35462 1/20 0.47
CYP3A4 P08684 1/20 0.46
HSD17B10 Q99714 1/20 0.46
KCNH2 Q12809 1/20 0.46
CCR3 P51677 1/20 0.45
KMT2A Q03164 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8555562 0.84 DRD4 (0.54) SIGMAR1ALDH1A1DRD4LMNADRD2
SCHEMBL8555816 0.83 SIGMAR1 (0.56) SIGMAR1ALDH1A1DRD4KMT2A
SCHEMBL8558370 0.79 ALDH1A1 (0.53) SIGMAR1ALDH1A1LMNADRD2DRD3
SCHEMBL7481150 0.78 ALDH1A1 (0.41) ALDH1A1POLBKMT2A
SCHEMBL8558421 0.78 ALDH1A1 (0.55) SIGMAR1ALDH1A1DRD4POLBLMNA
SCHEMBL8560914 0.78 KCNH2 (0.55) ALDH1A1DRD4LMNADRD2DRD3
SCHEMBL2489199 0.76 SIGMAR1 (1.00) SIGMAR1MC4RDRD4POLBLMNA
SCHEMBL576868 0.76 SIGMAR1 (1.00) SIGMAR1MC4RDRD4POLBLMNA
SCHEMBL8188324 0.76 SIGMAR1 (1.00) SIGMAR1MC4RDRD4POLBLMNA
SCHEMBL1415730 0.76 SIGMAR1 (1.00) SIGMAR1MC4RDRD4POLBLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0883622-A1 PROTON PUMP INHIBITOR APOTEX INC. (CA) 1998-12-16 EP claimed
WO-1997031923-A1 PROTON PUMP INHIBITOR APOTEX INC. (CA) 1997-09-04 WO claimed
EP-0883622-A1 PROTON PUMP INHIBITOR APOTEX INC. (CA) 1998-12-16 EP disclosed
EP-0883606-A1 PROCESS FOR SCAVENGING THIOLS APOTEX INC. (CA) 1998-12-16 EP disclosed
WO-1997031923-A1 PROTON PUMP INHIBITOR APOTEX INC. (CA) 1997-09-04 WO disclosed
WO-1997031893-A1 PROCESS FOR SCAVENGING THIOLS APOTEX INC. (CA) 1997-09-04 WO disclosed